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1.
Synthesis and structure-activity relationships of ticlopidine derivatives and analogs as inhibitors of ectonucleotidase CD39.
Bioorg Chem
; 135: 106460, 2023 06.
Artículo
en Inglés
| MEDLINE | ID: mdl-37023582
2.
Sulfated Polysaccharides from Macroalgae Are Potent Dual Inhibitors of Human ATP-Hydrolyzing Ectonucleotidases NPP1 and CD39.
Mar Drugs
; 19(2)2021 Jan 22.
Artículo
en Inglés
| MEDLINE | ID: mdl-33499103
3.
2-Substituted thienotetrahydropyridine derivatives: Allosteric ectonucleotidase inhibitors.
Arch Pharm (Weinheim)
; 354(12): e2100300, 2021 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-34697820
4.
Targeting the Main Protease of SARS-CoV-2: From the Establishment of High Throughput Screening to the Design of Tailored Inhibitors.
Angew Chem Int Ed Engl
; 60(18): 10423-10429, 2021 04 26.
Artículo
en Inglés
| MEDLINE | ID: mdl-33655614
5.
Correction to "Cathepsin-Targeting SARS-CoV-2 Inhibitors: Design, Synthesis, and Biological Activity".
ACS Pharmacol Transl Sci
; 7(4): 1195-1196, 2024 Apr 12.
Artículo
en Inglés
| MEDLINE | ID: mdl-38633592
6.
Cathepsin-Targeting SARS-CoV-2 Inhibitors: Design, Synthesis, and Biological Activity.
ACS Pharmacol Transl Sci
; 7(2): 493-514, 2024 Feb 09.
Artículo
en Inglés
| MEDLINE | ID: mdl-38357286
7.
Heparins are potent inhibitors of ectonucleotide pyrophosphatase/phospho-diesterase-1 (NPP1) - a promising target for the immunotherapy of cancer.
Front Immunol
; 14: 1173634, 2023.
Artículo
en Inglés
| MEDLINE | ID: mdl-37711611
8.
Protein kinase inhibitor ceritinib blocks ectonucleotidase CD39 - a promising target for cancer immunotherapy.
J Immunother Cancer
; 10(8)2022 08.
Artículo
en Inglés
| MEDLINE | ID: mdl-35981785
9.
Discovery and Crystallographic Studies of Nonpeptidic Piperazine Derivatives as Covalent SARS-CoV-2 Main Protease Inhibitors.
J Med Chem
; 65(24): 16902-16917, 2022 12 22.
Artículo
en Inglés
| MEDLINE | ID: mdl-36475694
10.
3CL Protease Inhibitors with an Electrophilic Arylketone Moiety as Anti-SARS-CoV-2 Agents.
J Med Chem
; 65(4): 2926-2939, 2022 02 24.
Artículo
en Inglés
| MEDLINE | ID: mdl-34313428
11.
Discovery and Crystallographic Studies of Trisubstituted Piperazine Derivatives as Non-Covalent SARS-CoV-2 Main Protease Inhibitors with High Target Specificity and Low Toxicity.
J Med Chem
; 65(19): 13343-13364, 2022 10 13.
Artículo
en Inglés
| MEDLINE | ID: mdl-36107752
12.
Small-Molecule Thioesters as SARS-CoV-2 Main Protease Inhibitors: Enzyme Inhibition, Structure-Activity Relationships, Antiviral Activity, and X-ray Structure Determination.
J Med Chem
; 65(13): 9376-9395, 2022 07 14.
Artículo
en Inglés
| MEDLINE | ID: mdl-35709506
13.
Development of Anthraquinone Derivatives as Ectonucleoside Triphosphate Diphosphohydrolase (NTPDase) Inhibitors With Selectivity for NTPDase2 and NTPDase3.
Front Pharmacol
; 11: 1282, 2020.
Artículo
en Inglés
| MEDLINE | ID: mdl-32973513
14.
Nucleotide Analog ARL67156 as a Lead Structure for the Development of CD39 and Dual CD39/CD73 Ectonucleotidase Inhibitors.
Front Pharmacol
; 11: 1294, 2020.
Artículo
en Inglés
| MEDLINE | ID: mdl-33013365
15.
Fluorescent Probes for Ecto-5'-nucleotidase (CD73).
ACS Med Chem Lett
; 11(11): 2253-2260, 2020 Nov 12.
Artículo
en Inglés
| MEDLINE | ID: mdl-33214837
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