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1.
Design, synthesis, and pharmacological profiling of cannabinoid 1 receptor allosteric modulators: Preclinical efficacy of C2-group GAT211 congeners for reducing intraocular pressure.
Bioorg Med Chem
; 50: 116421, 2021 11 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-34634617
2.
Focused structure-activity relationship profiling around the 2-phenylindole scaffold of a cannabinoid type-1 receptor agonist-positive allosteric modulator: site-III aromatic-ring congeners with enhanced activity and solubility.
Bioorg Med Chem
; 28(21): 115727, 2020 11 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-33065437
3.
Discovery of a Biased Allosteric Modulator for Cannabinoid 1 Receptor: Preclinical Anti-Glaucoma Efficacy.
J Med Chem
; 64(12): 8104-8126, 2021 06 24.
Artículo
en Inglés
| MEDLINE | ID: mdl-33826336
4.
Application of Fluorine- and Nitrogen-Walk Approaches: Defining the Structural and Functional Diversity of 2-Phenylindole Class of Cannabinoid 1 Receptor Positive Allosteric Modulators.
J Med Chem
; 63(2): 542-568, 2020 01 23.
Artículo
en Inglés
| MEDLINE | ID: mdl-31756109
5.
Identification of CB1 Receptor Allosteric Sites Using Force-Biased MMC Simulated Annealing and Validation by Structure-Activity Relationship Studies.
ACS Med Chem Lett
; 10(8): 1216-1221, 2019 Aug 08.
Artículo
en Inglés
| MEDLINE | ID: mdl-31413808
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