Detalles de la búsqueda
1.
EGCG Disrupts the LIN28B/Let-7 Interaction and Reduces Neuroblastoma Aggressiveness.
Int J Mol Sci
; 25(9)2024 Apr 27.
Artículo
en Inglés
| MEDLINE | ID: mdl-38732012
2.
α-Glucosidase inhibition by green, white and oolong teas: in vitro activity and computational studies.
J Enzyme Inhib Med Chem
; 38(1): 2236802, 2023 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-37470394
3.
Synthesis, in silico modelling, and in vitro biological evaluation of substituted pyrazole derivatives as potential anti-skin cancer, anti-tyrosinase, and antioxidant agents.
J Enzyme Inhib Med Chem
; 38(1): 2205042, 2023 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-37184042
4.
Synthesis, inverse docking-assisted identification and in vitro biological characterization of Flavonol-based analogs of fisetin as c-Kit, CDK2 and mTOR inhibitors against melanoma and non-melanoma skin cancers.
Bioorg Chem
; 107: 104595, 2021 02.
Artículo
en Inglés
| MEDLINE | ID: mdl-33450548
5.
Proproliferative function of adaptor protein GRB10 in prostate carcinoma.
FASEB J
; 33(3): 3198-3211, 2019 03.
Artículo
en Inglés
| MEDLINE | ID: mdl-30379590
6.
Inhibitory Effect of 2,3,5,6-Tetrafluoro-4-[4-(aryl)-1H-1,2,3-triazol-1-yl]benzenesulfonamide Derivatives on HIV Reverse Transcriptase Associated RNase H Activities.
Int J Mol Sci
; 17(8)2016 Aug 20.
Artículo
en Inglés
| MEDLINE | ID: mdl-27556447
7.
An integrated biological approach to guide the development of metal-chelating inhibitors of influenza virus PA endonuclease.
Mol Pharmacol
; 87(2): 323-37, 2015 Feb.
Artículo
en Inglés
| MEDLINE | ID: mdl-25477342
8.
Design and discovery of novel quinazolinedione-based redox modulators as therapies for pancreatic cancer.
Biochim Biophys Acta
; 1840(1): 332-43, 2014 Jan.
Artículo
en Inglés
| MEDLINE | ID: mdl-23954204
9.
Investigation of the salicylaldehyde thiosemicarbazone scaffold for inhibition of influenza virus PA endonuclease.
J Biol Inorg Chem
; 20(7): 1109-21, 2015 Oct.
Artículo
en Inglés
| MEDLINE | ID: mdl-26323352
10.
Peptidomimetics as protein arginine deiminase 4 (PAD4) inhibitors.
J Enzyme Inhib Med Chem
; 30(3): 466-71, 2015 Jun.
Artículo
en Inglés
| MEDLINE | ID: mdl-25198885
11.
Mutational analysis of the binding pockets of the diketo acid inhibitor L-742,001 in the influenza virus PA endonuclease.
J Virol
; 87(19): 10524-38, 2013 Oct.
Artículo
en Inglés
| MEDLINE | ID: mdl-23824822
12.
Metal-chelating 2-hydroxyphenyl amide pharmacophore for inhibition of influenza virus endonuclease.
Mol Pharm
; 11(1): 304-16, 2014 Jan 06.
Artículo
en Inglés
| MEDLINE | ID: mdl-24206028
13.
Resveratrol-loaded nanoparticles based on poly(epsilon-caprolactone) and poly(D,L-lactic-co-glycolic acid)-poly(ethylene glycol) blend for prostate cancer treatment.
Mol Pharm
; 10(10): 3871-81, 2013 Oct 07.
Artículo
en Inglés
| MEDLINE | ID: mdl-23968375
14.
Inhibition of α-class cytosolic human carbonic anhydrases I, II, IX and XII, and ß-class fungal enzymes by carboxylic acids and their derivatives: new isoform-I selective nanomolar inhibitors.
Bioorg Med Chem Lett
; 22(18): 5801-6, 2012 Sep 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-22901388
15.
Nanoparticle therapeutics for prostate cancer treatment.
Nanomedicine
; 8 Suppl 1: S31-6, 2012 Sep.
Artículo
en Inglés
| MEDLINE | ID: mdl-22640911
16.
Development of targeted nanoparticles loaded with antiviral drugs for SARS-CoV-2 inhibition.
Eur J Med Chem
; 231: 114121, 2022 Mar 05.
Artículo
en Inglés
| MEDLINE | ID: mdl-35114539
17.
HIV-1 IN strand transfer chelating inhibitors: a focus on metal binding.
Mol Pharm
; 8(2): 507-19, 2011 Apr 04.
Artículo
en Inglés
| MEDLINE | ID: mdl-21323359
18.
Development of polymeric microbubbles targeted to prostate-specific membrane antigen as prototype of novel ultrasound contrast agents.
Mol Pharm
; 8(3): 748-57, 2011 Jun 06.
Artículo
en Inglés
| MEDLINE | ID: mdl-21545176
19.
Virtual screening-driven identification of human carbonic anhydrase inhibitors incorporating an original, new pharmacophore.
Bioorg Med Chem Lett
; 21(8): 2515-20, 2011 Apr 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-21420862
20.
Identification of new fisetin analogs as kinase inhibitors: Data on synthesis and anti-skin cancer activities evaluation.
Data Brief
; 35: 106858, 2021 Apr.
Artículo
en Inglés
| MEDLINE | ID: mdl-33665254