Detalles de la búsqueda
1.
Synthesis, In Silico and Kinetics Evaluation of N-(ß-d-glucopyranosyl)-2-arylimidazole-4(5)-carboxamides and N-(ß-d-glucopyranosyl)-4(5)-arylimidazole-2-carboxamides as Glycogen Phosphorylase Inhibitors.
Int J Mol Sci
; 25(9)2024 Apr 23.
Artículo
en Inglés
| MEDLINE | ID: mdl-38731811
2.
Design and Synthesis of 3-(ß-d-Glucopyranosyl)-4-amino/4-guanidino Pyrazole Derivatives and Analysis of Their Glycogen Phosphorylase Inhibitory Potential.
Molecules
; 28(7)2023 Mar 28.
Artículo
en Inglés
| MEDLINE | ID: mdl-37049768
3.
Half-Sandwich Type Platinum-Group Metal Complexes of C-Glucosaminyl Azines: Synthesis and Antineoplastic and Antimicrobial Activities.
Molecules
; 28(7)2023 Mar 29.
Artículo
en Inglés
| MEDLINE | ID: mdl-37049820
4.
Reactive Oxygen Species Production Is Responsible for Antineoplastic Activity of Osmium, Ruthenium, Iridium and Rhodium Half-Sandwich Type Complexes with Bidentate Glycosyl Heterocyclic Ligands in Various Cancer Cell Models.
Int J Mol Sci
; 23(2)2022 Jan 12.
Artículo
en Inglés
| MEDLINE | ID: mdl-35054999
5.
2-Acetamido-2-deoxy-d-glucono-1,5-lactone Sulfonylhydrazones: Synthesis and Evaluation as Inhibitors of Human OGA and HexB Enzymes.
Int J Mol Sci
; 23(3)2022 Jan 18.
Artículo
en Inglés
| MEDLINE | ID: mdl-35162960
6.
Glycopyranosylidene-Spiro-Morpholinones: Evaluation of the Synthetic Possibilities Based on Glyculosonamide Derivatives and a New Method for the Construction of the Morpholine Ring.
Molecules
; 27(22)2022 Nov 11.
Artículo
en Inglés
| MEDLINE | ID: mdl-36431884
7.
Coupling Reactions of Anhydro-Aldose Tosylhydrazones with Boronic Acids.
Molecules
; 27(6)2022 Mar 09.
Artículo
en Inglés
| MEDLINE | ID: mdl-35335162
8.
First Synthesis of 3-Glycopyranosyl-1,2,4-Triazines and Some Cycloadditions Thereof.
Molecules
; 27(22)2022 Nov 12.
Artículo
en Inglés
| MEDLINE | ID: mdl-36431902
9.
Coupling of N-tosylhydrazones with tetrazoles: synthesis of 2-ß-D-glycopyranosylmethyl-5-substituted-2H-tetrazole type glycomimetics.
Org Biomol Chem
; 19(3): 605-618, 2021 01 28.
Artículo
en Inglés
| MEDLINE | ID: mdl-33355586
10.
Ruthenium Half-Sandwich Type Complexes with Bidentate Monosaccharide Ligands Show Antineoplastic Activity in Ovarian Cancer Cell Models through Reactive Oxygen Species Production.
Int J Mol Sci
; 22(19)2021 Sep 28.
Artículo
en Inglés
| MEDLINE | ID: mdl-34638791
11.
Glucose-based spiro-oxathiazoles as in vivo anti-hyperglycemic agents through glycogen phosphorylase inhibition.
Org Biomol Chem
; 18(5): 931-940, 2020 02 07.
Artículo
en Inglés
| MEDLINE | ID: mdl-31922157
12.
The architecture of hydrogen and sulfur σ-hole interactions explain differences in the inhibitory potency of C-ß-d-glucopyranosyl thiazoles, imidazoles and an N-ß-d glucopyranosyl tetrazole for human liver glycogen phosphorylase and offer new insights to structure-based design.
Bioorg Med Chem
; 28(1): 115196, 2020 01 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-31767404
13.
Stereoselective Synthesis of Carbon-Sulfur-Bridged Glycomimetics by Photoinitiated Thiol-Ene Coupling Reactions.
Int J Mol Sci
; 21(2)2020 Jan 16.
Artículo
en Inglés
| MEDLINE | ID: mdl-31963149
14.
Synthesis of New Series of 2-C-(ß-D-glucopyranosyl)-Pyrimidines and Their Evaluation as Inhibitors of Some Glycoenzymes.
Molecules
; 25(3)2020 Feb 06.
Artículo
en Inglés
| MEDLINE | ID: mdl-32041285
15.
C-Glycopyranosyl Arenes and Hetarenes: Synthetic Methods and Bioactivity Focused on Antidiabetic Potential.
Chem Rev
; 117(3): 1687-1764, 2017 02 08.
Artículo
en Inglés
| MEDLINE | ID: mdl-28121130
16.
Probing the ß-pocket of the active site of human liver glycogen phosphorylase with 3-(C-ß-d-glucopyranosyl)-5-(4-substituted-phenyl)-1, 2, 4-triazole inhibitors.
Bioorg Chem
; 77: 485-493, 2018 04.
Artículo
en Inglés
| MEDLINE | ID: mdl-29454281
17.
Synthesis of New C- and N-ß-d-Glucopyranosyl Derivatives of Imidazole, 1,2,3-Triazole and Tetrazole, and Their Evaluation as Inhibitors of Glycogen Phosphorylase.
Molecules
; 23(3)2018 Mar 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-29543771
18.
van der Waals interactions govern C-ß-d-glucopyranosyl triazoles' nM inhibitory potency in human liver glycogen phosphorylase.
J Struct Biol
; 199(1): 57-67, 2017 07.
Artículo
en Inglés
| MEDLINE | ID: mdl-28483603
19.
Glucopyranosylidene-Spiro-Thiazolinones: Synthetic Studies and Determination of Absolute Configuration by TDDFT-ECD Calculations.
Molecules
; 22(10)2017 Oct 19.
Artículo
en Inglés
| MEDLINE | ID: mdl-29048398
20.
Decomposition of N-chloroglycine in alkaline aqueous solution: kinetics and mechanism.
Chem Res Toxicol
; 28(6): 1282-91, 2015 Jun 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-25849302