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1.
Investigation of C-5 alkynyl (alkynyloxy or hydroxymethyl) and/or N-3 propynyl substituted pyrimidine nucleoside analogs as a new class of antimicrobial agents.
Bioorg Med Chem
; 24(21): 5521-5533, 2016 11 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-27665179
2.
Antimycobacterial activities of 5-alkyl (or halo)-3'-substituted pyrimidine nucleoside analogs.
Bioorg Med Chem Lett
; 22(2): 1091-4, 2012 Jan 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-22178557
3.
Discovery of novel 5-(ethyl or hydroxymethyl) analogs of 2'-'up' fluoro (or hydroxyl) pyrimidine nucleosides as a new class of Mycobacterium tuberculosis, Mycobacterium bovis and Mycobacterium avium inhibitors.
Bioorg Med Chem
; 20(13): 4088-97, 2012 Jul 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-22664188
4.
Antiviral activity of 2,3'-anhydro and related pyrimidine nucleosides against hepatitis B virus.
Bioorg Med Chem Lett
; 20(22): 6790-3, 2010 Nov 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-20863701
5.
Synthesis and in vitro antiviral activities of 3'-fluoro (or chloro) and 2',3'-difluoro 2',3'-dideoxynucleoside analogs against hepatitis B and C viruses.
Bioorg Med Chem
; 18(21): 7542-7, 2010 Nov 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-20869253
6.
Inhibition of Mycobacterium tuberculosis, Mycobacterium bovis, and Mycobacterium avium by novel dideoxy nucleosides.
J Med Chem
; 50(19): 4766-74, 2007 Sep 20.
Artículo
en Inglés
| MEDLINE | ID: mdl-17696514
7.
In vitro anti-mycobacterial activities of various 2'-deoxyuridine, 2'-arabinouridine and 2'-arabinofluoro-2'-deoxyuridine analogues: synthesis and biological studies.
Med Chem
; 2(3): 287-93, 2006 May.
Artículo
en Inglés
| MEDLINE | ID: mdl-16948475
8.
Inhibition of mycobacterial replication by pyrimidines possessing various C-5 functionalities and related 2'-deoxynucleoside analogues using in vitro and in vivo models.
J Med Chem
; 53(16): 6180-7, 2010 Aug 26.
Artículo
en Inglés
| MEDLINE | ID: mdl-20718497
9.
Antiviral activity of various 1-(2'-deoxy-ß-D-lyxofuranosyl), 1-(2'-fluoro-ß-D-xylofuranosyl), 1-(3'-fluoro-ß-D-arabinofuranosyl), and 2'-fluoro-2',3'-didehydro-2',3'-dideoxyribose pyrimidine nucleoside analogues against duck hepatitis B virus (DHBV) and human hepatitis B virus (HBV) replication.
J Med Chem
; 53(19): 7156-66, 2010 Oct 14.
Artículo
en Inglés
| MEDLINE | ID: mdl-20857959
10.
3'-bromo analogues of pyrimidine nucleosides as a new class of potent inhibitors of Mycobacterium tuberculosis.
J Med Chem
; 53(10): 4130-40, 2010 May 27.
Artículo
en Inglés
| MEDLINE | ID: mdl-20420370
11.
Studies on acyclic pyrimidines as inhibitors of mycobacteria.
Bioorg Med Chem
; 15(5): 2045-53, 2007 Mar 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-17218105
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