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1.
A knowledge-based, structural-aided discovery of a novel class of 2-phenylimidazo[1,2-a]pyridine-6-carboxamide H-PGDS inhibitors.
Bioorg Med Chem Lett
; 47: 128113, 2021 09 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-33991628
2.
The exploration of aza-quinolines as hematopoietic prostaglandin D synthase (H-PGDS) inhibitors with low brain exposure.
Bioorg Med Chem
; 28(23): 115791, 2020 12 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-33059303
3.
The discovery of quinoline-3-carboxamides as hematopoietic prostaglandin D synthase (H-PGDS) inhibitors.
Bioorg Med Chem
; 27(8): 1456-1478, 2019 04 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-30858025
4.
2,4-Diamino-8-quinazoline carboxamides as novel, potent inhibitors of the NAD hydrolyzing enzyme CD38: Exploration of the 2-position structure-activity relationships.
Bioorg Med Chem
; 26(8): 2107-2150, 2018 05 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-29576271
5.
Biochemical characterization of GSK1070916, a potent and selective inhibitor of Aurora B and Aurora C kinases with an extremely long residence time1.
Biochem J
; 420(2): 259-65, 2009 May 13.
Artículo
en Inglés
| MEDLINE | ID: mdl-19284385
6.
SIRT4 Is a Lysine Deacylase that Controls Leucine Metabolism and Insulin Secretion.
Cell Metab
; 25(4): 838-855.e15, 2017 Apr 04.
Artículo
en Inglés
| MEDLINE | ID: mdl-28380376
7.
Discovery of 4-Amino-8-quinoline Carboxamides as Novel, Submicromolar Inhibitors of NAD-Hydrolyzing Enzyme CD38.
J Med Chem
; 58(17): 7021-56, 2015 Sep 10.
Artículo
en Inglés
| MEDLINE | ID: mdl-26267483
8.
Discovery, Synthesis, and Biological Evaluation of Thiazoloquin(az)olin(on)es as Potent CD38 Inhibitors.
J Med Chem
; 58(8): 3548-71, 2015 Apr 23.
Artículo
en Inglés
| MEDLINE | ID: mdl-25828863
9.
Design and effective synthesis of novel templates, 3,7-diphenyl-4-amino-thieno and furo-[3,2-c]pyridines as protein kinase inhibitors and in vitro evaluation targeting angiogenetic kinases.
Bioorg Med Chem Lett
; 17(1): 250-4, 2007 Jan 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-17027260
10.
Comparison of the biochemical and kinetic properties of the type 1 receptor tyrosine kinase intracellular domains. Demonstration of differential sensitivity to kinase inhibitors.
J Biol Chem
; 277(2): 1576-85, 2002 Jan 11.
Artículo
en Inglés
| MEDLINE | ID: mdl-11696537
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