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1.
Discovery of 3-hydroxymethyl-azetidine derivatives as potent polymerase theta inhibitors.
Bioorg Med Chem
; 103: 117662, 2024 Apr 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-38493730
2.
Discovery and preclinical profile of LX-039, a novel indole-based oral selective estrogen receptor degrader (SERD).
Bioorg Med Chem Lett
; 66: 128734, 2022 06 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-35436589
3.
Design, syntheses and evaluations of novel indole derivatives as orally selective estrogen receptor degraders (SERD).
Bioorg Med Chem Lett
; 30(22): 127601, 2020 11 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-33035677
4.
Highly Selective Fluorescent Turn-On Probe for Protein Thiols in Biotin Receptor-Positive Cancer Cells.
Anal Chem
; 88(6): 3400-5, 2016 Mar 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-26902836
5.
Discrimination between streptavidin and avidin with fluorescent affinity-based probes.
Analyst
; 140(13): 4648-53, 2015 Jul 07.
Artículo
en Inglés
| MEDLINE | ID: mdl-25985268
6.
Antiproliferative and apoptosis-inducing activities of novel naphthalimide-cyclam conjugates through dual topoisomerase (topo) I/II inhibition.
Bioorg Med Chem
; 23(17): 5672-80, 2015 Sep 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-26211460
7.
Synthesis and structure-activity optimization of azepane-containing derivatives as PTPN2/PTPN1 inhibitors.
Eur J Med Chem
; 270: 116390, 2024 Apr 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-38604096
8.
Recent progress in silk fibroin-based flexible electronics.
Microsyst Nanoeng
; 7: 35, 2021.
Artículo
en Inglés
| MEDLINE | ID: mdl-34567749
9.
Discovery of Potent and Noncovalent Reversible EGFR Kinase Inhibitors of EGFRL858R/T790M/C797S.
ACS Med Chem Lett
; 10(6): 869-873, 2019 Jun 13.
Artículo
en Inglés
| MEDLINE | ID: mdl-31223440
10.
Design, Synthesis, and Biological Evaluation of Pyrimido[4,5- d]pyrimidine-2,4(1 H,3 H)-diones as Potent and Selective Epidermal Growth Factor Receptor (EGFR) Inhibitors against L858R/T790M Resistance Mutation.
J Med Chem
; 61(13): 5609-5622, 2018 07 12.
Artículo
en Inglés
| MEDLINE | ID: mdl-29906114
11.
Structure-Guided Design of C4-alkyl-1,4-dihydro-2H-pyrimido[4,5-d][1,3]oxazin-2-ones as Potent and Mutant-Selective Epidermal Growth Factor Receptor (EGFR) L858R/T790M Inhibitors.
Sci Rep
; 7(1): 3830, 2017 06 19.
Artículo
en Inglés
| MEDLINE | ID: mdl-28630494
12.
Discovery and Rational Design of Pteridin-7(8H)-one-Based Inhibitors Targeting FMS-like Tyrosine Kinase 3 (FLT3) and Its Mutants.
J Med Chem
; 59(13): 6187-200, 2016 07 14.
Artículo
en Inglés
| MEDLINE | ID: mdl-27266526
13.
Carbazole Aminoalcohols Induce Antiproliferation and Apoptosis of Human Tumor Cells by Inhibiting Topoisomeraseâ I.
ChemMedChem
; 11(24): 2675-2681, 2016 12 16.
Artículo
en Inglés
| MEDLINE | ID: mdl-27879063
14.
Discovery and Structural Optimization of N5-Substituted 6,7-Dioxo-6,7-dihydropteridines as Potent and Selective Epidermal Growth Factor Receptor (EGFR) Inhibitors against L858R/T790M Resistance Mutation.
J Med Chem
; 59(15): 7111-24, 2016 08 11.
Artículo
en Inglés
| MEDLINE | ID: mdl-27396610
15.
Novel selective and potent inhibitors of malaria parasite dihydroorotate dehydrogenase: discovery and optimization of dihydrothiophenone derivatives.
J Med Chem
; 56(20): 7911-24, 2013 Oct 24.
Artículo
en Inglés
| MEDLINE | ID: mdl-24073986
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