Detalles de la búsqueda
1.
Design and synthesis of trans-N-[4-[2-(6-cyano-1,2,3, 4-tetrahydroisoquinolin-2-yl)ethyl]cyclohexyl]-4-quinolinecarboxamide (SB-277011): A potent and selective dopamine D(3) receptor antagonist with high oral bioavailability and CNS penetration in the rat.
J Med Chem
; 43(9): 1878-85, 2000 May 04.
Artículo
en Inglés
| MEDLINE | ID: mdl-10794704
2.
Novel and selective 5-HT2C/2B receptor antagonists as potential anxiolytic agents: synthesis, quantitative structure-activity relationships, and molecular modeling of substituted 1-(3-pyridylcarbamoyl)indolines.
J Med Chem
; 41(10): 1598-612, 1998 May 07.
Artículo
en Inglés
| MEDLINE | ID: mdl-9572885
3.
6-Chloro-5-methyl-1-[[2-[(2-methyl-3-pyridyl)oxy]-5-pyridyl]carbamoyl]- indoline (SB-242084): the first selective and brain penetrant 5-HT2C receptor antagonist.
J Med Chem
; 40(22): 3494-6, 1997 Oct 24.
Artículo
en Inglés
| MEDLINE | ID: mdl-9357513
4.
Novel 2,3,4,5-tetrahydro-1H-3-benzazepines with high affinity and selectivity for the dopamine D3 receptor.
Bioorg Med Chem Lett
; 10(22): 2553-5, 2000 Nov 20.
Artículo
en Inglés
| MEDLINE | ID: mdl-11086728
5.
Fused aminotetralins: novel antagonists with high selectivity for the dopamine D3 receptor.
Bioorg Med Chem Lett
; 8(20): 2859-64, 1998 Oct 20.
Artículo
en Inglés
| MEDLINE | ID: mdl-9873637
6.
Novel 1,2,3,4-tetrahydroisoquinolines with high affinity and selectivity for the dopamine D3 receptor.
Bioorg Med Chem Lett
; 9(2): 179-84, 1999 Jan 18.
Artículo
en Inglés
| MEDLINE | ID: mdl-10021923
7.
Model studies on a synthetically facile series of N-substituted phenyl-N'-pyridin-3-yl ureas leading to 1-(3-pyridylcarbamoyl) indolines that are potent and selective 5-HT(2C/2B) receptor antagonists.
Bioorg Med Chem
; 7(12): 2767-73, 1999 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-10658582
8.
Design and synthesis of novel 2,3-dihydro-1H-isoindoles with high affinity and selectivity for the dopamine D3 receptor.
Bioorg Med Chem Lett
; 11(5): 685-8, 2001 Mar 12.
Artículo
en Inglés
| MEDLINE | ID: mdl-11266169
9.
Pharmacological actions of a novel, high-affinity, and selective human dopamine D(3) receptor antagonist, SB-277011-A.
J Pharmacol Exp Ther
; 294(3): 1154-65, 2000 Sep.
Artículo
en Inglés
| MEDLINE | ID: mdl-10945872
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