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1.
Design, synthesis and validation of a new Crimped Head-Piece for DNA-Encoded libraries generation.
Bioorg Med Chem
; 99: 117596, 2024 Feb 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-38232459
2.
On-DNA Palladium-Catalyzed Hydrogenation-like Reaction Suitable for DNA-Encoded Library Synthesis.
Bioconjug Chem
; 32(1): 88-93, 2021 01 20.
Artículo
en Inglés
| MEDLINE | ID: mdl-33356163
3.
Enantioselective Synthesis of 3,3-Difluoropyrrolidin-4-ol, a Valuable Building Block in Medicinal Chemistry.
J Org Chem
; 81(10): 4359-63, 2016 05 20.
Artículo
en Inglés
| MEDLINE | ID: mdl-27138111
4.
Competing thermal electrocyclic ring-closure reactions of (2Z)-hexa-2,4,5-trienals and their Schiff bases. Structural, kinetic, and computational studies.
J Org Chem
; 75(13): 4453-62, 2010 Jul 02.
Artículo
en Inglés
| MEDLINE | ID: mdl-20521841
5.
Mild and Efficient Palladium-Mediated C-N Cross-Coupling Reaction between DNA-Conjugated Aryl Bromides and Aromatic Amines.
ACS Comb Sci
; 21(2): 69-74, 2019 02 11.
Artículo
en Inglés
| MEDLINE | ID: mdl-30615417
6.
Characterization of a novel AICARFT inhibitor which potently elevates ZMP and has anti-tumor activity in murine models.
Sci Rep
; 8(1): 15458, 2018 10 18.
Artículo
en Inglés
| MEDLINE | ID: mdl-30337562
7.
Discovery of N-(6-Fluoro-1-oxo-1,2-dihydroisoquinolin-7-yl)-5-[(3R)-3-hydroxypyrrolidin-1-yl]thiophene-2-sulfonamide (LSN 3213128), a Potent and Selective Nonclassical Antifolate Aminoimidazole-4-carboxamide Ribonucleotide Formyltransferase (AICARFT) Inhibitor Effective at Tumor Suppression in a Cancer Xenograft Model.
J Med Chem
; 60(23): 9599-9616, 2017 12 14.
Artículo
en Inglés
| MEDLINE | ID: mdl-29072452
8.
New Synthetic Amino Acids for the Design and Synthesis of Peptide-Based Metal Ion Sensors.
J Org Chem
; 61(25): 8940-8948, 1996 Dec 13.
Artículo
en Inglés
| MEDLINE | ID: mdl-11667875
9.
On the Aromatic Character of Electrocyclic and Pseudopericyclic Reactions: Thermal Cyclization of (2Z)-Hexa-2,4-5-trienals and Their Schiff Bases.
Angew Chem Int Ed Engl
; 40(3): 557-561, 2001 Feb 02.
Artículo
en Inglés
| MEDLINE | ID: mdl-29712011
10.
Discovery of a novel series of orally active nociceptin/orphanin FQ (NOP) receptor antagonists based on a dihydrospiro(piperidine-4,7'-thieno[2,3-c]pyran) scaffold.
J Med Chem
; 57(8): 3418-29, 2014 Apr 24.
Artículo
en Inglés
| MEDLINE | ID: mdl-24678969
11.
On the Aromatic Character of Electrocyclic and Pseudopericyclic Reactions: Thermal Cyclization of (2Z)-Hexa-2,4-5-trienals and Their Schiff Bases This work was supported by the Spanish Ministerio de Investigación (Grant no.: SAF98-0143), by the Xunta de Galicia (Grant no.: PGIDT99PXI30105B), by the Eusko Jaurlaritza (Grant nos.: EX1998-126 and PI1998-116), by Gipuzkoako Foru Aldundia, and by Fondo de Cooperación Aquitania-Euskadi. We thank Dr. J. Rodriguez-Otero and Dr. S. Lopez (Universidade de Santiago) for helpful discussions.
Angew Chem Int Ed Engl
; 40(3): 557-561, 2001 Feb 02.
Artículo
en Inglés
| MEDLINE | ID: mdl-11180369
12.
2-Alkoxydihydrocinnamates as PPAR agonists. Activity modulation by the incorporation of phenoxy substituents.
Bioorg Med Chem Lett
; 15(1): 51-5, 2005 Jan 03.
Artículo
en Inglés
| MEDLINE | ID: mdl-15582409
13.
Stereoselective synthesis of annular 9-cis-retinoids and binding characterization to the retinoid X receptor.
J Org Chem
; 67(17): 5876-82, 2002 Aug 23.
Artículo
en Inglés
| MEDLINE | ID: mdl-12182616
14.
Novel selective and potent 5-HT reuptake inhibitors with 5-HT1D antagonist activity: chemistry and pharmacological evaluation of a series of thienopyran derivatives.
Bioorg Med Chem
; 12(20): 5277-95, 2004 Oct 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-15388156
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