Detalles de la búsqueda
1.
Investigations on substituted (2-aminothiazol-5-yl)(imidazo[1,2-a]pyridin-3-yl)methanones for the treatment of Alzheimer's disease.
Bioorg Med Chem
; 36: 116091, 2021 04 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-33676335
2.
Pharmacological investigation of quinoxaline-bisthiazoles as multitarget-directed ligands for the treatment of Alzheimer's disease.
Bioorg Chem
; 89: 102992, 2019 08.
Artículo
en Inglés
| MEDLINE | ID: mdl-31174042
3.
Imidazo[1,2-a]pyridines linked with thiazoles/thiophene motif through keto spacer as potential cytotoxic agents and NF-κB inhibitors.
Bioorg Med Chem Lett
; 27(24): 5463-5466, 2017 12 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-29138027
4.
Design, synthesis and biological evaluation of novel pyrazolo-pyrimidinones as DPP-IV inhibitors in diabetes.
Bioorg Med Chem Lett
; 25(20): 4428-33, 2015 Oct 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-26372650
5.
Novel thiazole-thiophene conjugates as adenosine receptor antagonists: synthesis, biological evaluation and docking studies.
Bioorg Med Chem Lett
; 25(6): 1306-9, 2015 Mar 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-25686851
6.
Implication of novel thiazolo-thiophene derivative (MCD-KV-10) for management of asthma.
J Enzyme Inhib Med Chem
; 30(2): 229-39, 2015 Apr.
Artículo
en Inglés
| MEDLINE | ID: mdl-24939098
7.
Detoxification of Nerium indicum roots based on Indian system of medicine: phytochemical and toxicity evaluations.
Acta Pol Pharm
; 68(6): 905-11, 2011.
Artículo
en Inglés
| MEDLINE | ID: mdl-22125956
8.
Design, synthesis and evaluation of novel 2-thiophen-5-yl-3H-quinazolin-4-one analogues as inhibitors of transcription factors NF-kappaB and AP-1 mediated transcriptional activation: Their possible utilization as anti-inflammatory and anti-cancer agents.
Bioorg Med Chem
; 18(7): 2796-808, 2010 Apr 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-20335039
9.
2-Amino-5-benzoyl-4-phenylthiazoles: Development of potent and selective adenosine A1 receptor antagonists.
Bioorg Med Chem
; 18(6): 2195-2203, 2010 Mar 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-20188574
10.
Synthesis of 4-benzyl-1,3-thiazole derivatives as potential anti-inflammatory agents: an analogue-based drug design approach.
J Enzyme Inhib Med Chem
; 24(3): 890-7, 2009 Jun.
Artículo
en Inglés
| MEDLINE | ID: mdl-19469712
11.
Pair wise binding affinity: 3D QSAR studies on a set of triazolo [1, 5-a] quinoxalines as antagonists of AMPA and KA receptors.
J Enzyme Inhib Med Chem
; 24(4): 1008-14, 2009 Aug.
Artículo
en Inglés
| MEDLINE | ID: mdl-19548793
12.
2-Amino-5-thiazolyl motif: a novel scaffold for designing anti-inflammatory agents of diverse structures.
Eur J Med Chem
; 43(1): 129-34, 2008 Jan.
Artículo
en Inglés
| MEDLINE | ID: mdl-17467123
13.
Design, synthesis, and evaluation of 4,5,6,7-tetrahydrobenzo[d]thiazole-based novel dual kinase inhibitors of CK2 and GSK3ß.
Medchemcomm
; 9(9): 1472-1490, 2018 Sep 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-30288222
14.
Discovery of 2-aminoimidazole and 2-amino imidazolyl-thiazoles as non-xanthine human adenosine A3 receptor antagonists: SAR and molecular modeling studies.
Medchemcomm
; 9(4): 676-684, 2018 Apr 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-30108958
15.
Thiazolyl-thiadiazines as Beta Site Amyloid Precursor Protein Cleaving Enzyme-1 (BACE-1) Inhibitors and Anti-inflammatory Agents: Multitarget-Directed Ligands for the Efficient Management of Alzheimer's Disease.
ACS Chem Neurosci
; 9(7): 1663-1679, 2018 07 18.
Artículo
en Inglés
| MEDLINE | ID: mdl-29697965
16.
Syntheses of new tetrasubstituted thiophenes as novel anti-inflammatory agents.
Eur J Med Chem
; 42(8): 1049-58, 2007 Aug.
Artículo
en Inglés
| MEDLINE | ID: mdl-17336429
17.
Development and Validation of a Stability-Indicating HPLC Method for Imidapril and Its Degradation Products Using a Design of Experiment (DoE) Approach.
J AOAC Int
; 100(6): 1727-1738, 2017 Nov 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-28803600
18.
Impact of Ternary Solvent System in Stability-Indicating Assay Method of Bambuterol: Design of Experiments Approach.
J Chromatogr Sci
; 54(2): 221-9, 2016 Feb.
Artículo
en Inglés
| MEDLINE | ID: mdl-26362115
19.
In vivo Evaluation of Self Emulsifying Drug Delivery System for Oral Delivery of Nevirapine.
Indian J Pharm Sci
; 76(3): 218-24, 2014 May.
Artículo
en Inglés
| MEDLINE | ID: mdl-25035533
20.
Stability-indicating assay method for determination of actarit, its process related impurities and degradation products: Insight into stability profile and degradation pathwaysâ.
J Pharm Anal
; 4(6): 374-383, 2014 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-29403903