Detalles de la búsqueda
1.
Discovery of Conformationally Constrained ALK2 Inhibitors.
J Med Chem
; 67(6): 4707-4725, 2024 Mar 28.
Artículo
en Inglés
| MEDLINE | ID: mdl-38498998
2.
Triaryl (Z)-olefins suitable for radiolabeling with iodine-124 or fluorine-18 radionuclides for positron emission tomography imaging of estrogen positive breast tumors.
Bioorg Med Chem Lett
; 21(4): 1195-8, 2011 Feb 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-21237640
3.
Structure-Activity Relationship of USP5 Inhibitors.
J Med Chem
; 64(20): 15017-15036, 2021 10 28.
Artículo
en Inglés
| MEDLINE | ID: mdl-34648286
4.
A First-in-Class, Highly Selective and Cell-Active Allosteric Inhibitor of Protein Arginine Methyltransferase 6.
J Med Chem
; 64(7): 3697-3706, 2021 04 08.
Artículo
en Inglés
| MEDLINE | ID: mdl-33591753
5.
Comparison between 3-Nitrooxyphenyl acetylsalicylate (NO-ASA) and O2-(acetylsalicyloxymethyl)-1-(pyrrolidin-1-yl)diazen-1-ium-1,2-diolate (NONO-ASA) as safe anti-inflammatory, analgesic, antipyretic, antioxidant prodrugs.
J Pharmacol Exp Ther
; 335(2): 443-50, 2010 Nov.
Artículo
en Inglés
| MEDLINE | ID: mdl-20679133
6.
Triaryl (Z)-olefins suitable for radiolabeling with carbon-11 or fluorine-18 radionuclides for positron emission tomography imaging of cyclooxygenase-2 expression in pathological disease.
Bioorg Med Chem Lett
; 20(17): 5245-50, 2010 Sep 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-20655211
7.
Synthesis and biological evaluation of indomethacin analogs possessing a N-difluoromethyl-1,2-dihydropyrid-2-one ring system: a search for novel cyclooxygenase and lipoxygenase inhibitors.
Bioorg Med Chem Lett
; 20(19): 5776-80, 2010 Oct 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-20727750
8.
Celecoxib prodrugs possessing a diazen-1-ium-1,2-diolate nitric oxide donor moiety: synthesis, biological evaluation and nitric oxide release studies.
Bioorg Med Chem Lett
; 20(15): 4544-9, 2010 Aug 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-20576432
9.
Phenylacetic acid regioisomers possessing a N-difluoromethyl-1,2-dihydropyrid-2-one pharmacophore: evaluation as dual inhibitors of cyclooxygenases and 5-lipoxygenase with anti-inflammatory activity.
Bioorg Med Chem Lett
; 20(3): 896-902, 2010 Feb 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-20045320
10.
Celecoxib analogs possessing a N-(4-nitrooxybutyl)piperidin-4-yl or N-(4-nitrooxybutyl)-1,2,3,6-tetrahydropyridin-4-yl nitric oxide donor moiety: synthesis, biological evaluation and nitric oxide release studies.
Bioorg Med Chem Lett
; 20(4): 1324-9, 2010 Feb 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-20097072
11.
Synthesis and biological evaluation of N-difluoromethyl-1,2-dihydropyrid-2-one acetic acid regioisomers: dual inhibitors of cyclooxygenases and 5-lipoxygenase.
Bioorg Med Chem Lett
; 20(7): 2168-73, 2010 Apr 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-20202839
12.
Targeting ALK2: An Open Science Approach to Developing Therapeutics for the Treatment of Diffuse Intrinsic Pontine Glioma.
J Med Chem
; 63(9): 4978-4996, 2020 05 14.
Artículo
en Inglés
| MEDLINE | ID: mdl-32369358
13.
Dinitroglyceryl and diazen-1-ium-1,2-diolated nitric oxide donor ester prodrugs of aspirin, indomethacin and ibuprofen: synthesis, biological evaluation and nitric oxide release studies.
Bioorg Med Chem Lett
; 19(11): 3014-8, 2009 Jun 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-19419861
14.
Synthesis and biological evaluation of salicylic acid and N-acetyl-2-carboxybenzenesulfonamide regioisomers possessing a N-difluoromethyl-1,2-dihydropyrid-2-one pharmacophore: dual inhibitors of cyclooxygenases and 5-lipoxygenase with anti-inflammatory activity.
Bioorg Med Chem Lett
; 19(24): 6855-61, 2009 Dec 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-19884005
15.
A chemical biology toolbox to study protein methyltransferases and epigenetic signaling.
Nat Commun
; 10(1): 19, 2019 01 03.
Artículo
en Inglés
| MEDLINE | ID: mdl-30604761
16.
Second-generation aspirin and indomethacin prodrugs possessing an O(2)-(acetoxymethyl)-1-(2-carboxypyrrolidin-1-yl)diazenium-1,2-diolate nitric oxide donor moiety: design, synthesis, biological evaluation, and nitric oxide release studies.
J Med Chem
; 51(6): 1954-61, 2008 Mar 27.
Artículo
en Inglés
| MEDLINE | ID: mdl-18314945
17.
Técnica de la incisión y cierre de piel en "punto de mira" para la reversión de estoma. Experiencia en el Centro Médico Nacional "La Raza", México / Gunsight skin incision and closure technique for stoma reversal. Experience in Centro Médico Nacional "La Raza", México
Rev. argent. cir
; 115(2): 147-154, abr. 2023. graf
Artículo
en Español
|
LILACS-Express
| ID: biblio-1449390
18.
Correction to "Structure-Activity Relationship of USP5 Inhibitors".
J Med Chem
; 65(1): 889, 2022 Jan 13.
Artículo
en Inglés
| MEDLINE | ID: mdl-34958585
19.
Physical properties and antibacterial activity of chitosan/acemannan mixed systems.
Carbohydr Polym
; 115: 707-14, 2015 Jan 22.
Artículo
en Inglés
| MEDLINE | ID: mdl-25439952
20.
Ethanesulfohydroxamic acid ester prodrugs of nonsteroidal anti-inflammatory drugs (NSAIDs): synthesis, nitric oxide and nitroxyl release, cyclooxygenase inhibition, anti-inflammatory, and ulcerogenicity index studies.
J Med Chem
; 54(5): 1356-64, 2011 Mar 10.
Artículo
en Inglés
| MEDLINE | ID: mdl-21280601