Detalles de la búsqueda
1.
Rapid and Highly Selective Fluorescent Labeling of Peptides via a Thia-Diels-Alder Cycloaddition: Application to Apelin.
Bioconjug Chem
; 34(1): 162-168, 2023 01 18.
Artículo
en Inglés
| MEDLINE | ID: mdl-36534753
2.
Characterization of anti-GASP motif antibodies that inhibit the interaction between GPRASP1 and G protein-coupled receptors.
Anal Biochem
; 665: 115062, 2023 03 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-36731712
3.
Design, Synthesis and Biological Evaluation of Arylpyridin-2-yl Guanidine Derivatives and Cyclic Mimetics as Novel MSK1 Inhibitors. An Application in an Asthma Model.
Molecules
; 26(2)2021 Jan 13.
Artículo
en Inglés
| MEDLINE | ID: mdl-33450992
4.
Fluorogenic squaraine dimers with polarity-sensitive folding as bright far-red probes for background-free bioimaging.
J Am Chem Soc
; 137(1): 405-12, 2015 Jan 14.
Artículo
en Inglés
| MEDLINE | ID: mdl-25506627
5.
A general framework to characterize inhibitors of calmodulin: use of calmodulin inhibitors to study the interaction between calmodulin and its calmodulin binding domains.
Biochim Biophys Acta
; 1833(7): 1720-31, 2013 Jul.
Artículo
en Inglés
| MEDLINE | ID: mdl-23333870
6.
Red fluorescent turn-on ligands for imaging and quantifying G protein-coupled receptors in living cells.
Chembiochem
; 15(3): 359-63, 2014 Feb 10.
Artículo
en Inglés
| MEDLINE | ID: mdl-24449564
7.
Target-Focused Library Design by Pocket-Applied Computer Vision and Fragment Deep Generative Linking.
J Med Chem
; 65(20): 13771-13783, 2022 10 27.
Artículo
en Inglés
| MEDLINE | ID: mdl-36256484
8.
High-Throughput Screening for Extracellular Inhibitors of the FLT3 Receptor Tyrosine Kinase Reveals Chemically Diverse and Druggable Negative Allosteric Modulators.
ACS Chem Biol
; 17(3): 709-722, 2022 03 18.
Artículo
en Inglés
| MEDLINE | ID: mdl-35227060
9.
Treating leishmaniasis in Amazonia, part 2: Multi-target evaluation of widely used plants to understand medicinal practices.
J Ethnopharmacol
; 289: 115054, 2022 May 10.
Artículo
en Inglés
| MEDLINE | ID: mdl-35131338
10.
Antiallodynic action of phosphodiesterase inhibitors in a mouse model of peripheral nerve injury.
Neuropharmacology
; 205: 108909, 2022 03 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-34875284
11.
Engineering Novel 3D Models to Recreate High-Grade Osteosarcoma and its Immune and Extracellular Matrix Microenvironment.
Adv Healthc Mater
; 11(19): e2200195, 2022 10.
Artículo
en Inglés
| MEDLINE | ID: mdl-36057996
12.
Nile Red-Based GPCR Ligands as Ultrasensitive Probes of the Local Lipid Microenvironment of the Receptor.
ACS Chem Biol
; 16(4): 651-660, 2021 04 16.
Artículo
en Inglés
| MEDLINE | ID: mdl-33733725
13.
Overexpression of the MSK1 Kinase in Patients With Chronic Lung Allograft Dysfunction and Its Confirmed Role in a Murine Model.
Transplantation
; 105(6): 1212-1224, 2021 06 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-33560725
14.
Liposomal encapsulation of trans-crocetin enhances oxygenation in patients with COVID-19-related ARDS receiving mechanical ventilation.
J Control Release
; 336: 252-261, 2021 08 10.
Artículo
en Inglés
| MEDLINE | ID: mdl-34175365
15.
Identification by high-throughput screening of inhibitors of Schistosoma mansoni NAD(+) catabolizing enzyme.
Bioorg Med Chem
; 18(22): 7900-10, 2010 Nov 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-20951593
16.
Anti-Inflammatory, Antioxidant, and Wound-Healing Properties of Cyanobacteria from Thermal Mud of Balaruc-Les-Bains, France: A Multi-Approach Study.
Biomolecules
; 11(1)2020 12 29.
Artículo
en Inglés
| MEDLINE | ID: mdl-33383796
17.
Efficacy Assessment of an Uncharged Reactivator of NOP-Inhibited Acetylcholinesterase Based on Tetrahydroacridine Pyridine-Aldoxime Hybrid in Mouse Compared to Pralidoxime.
Biomolecules
; 10(6)2020 06 04.
Artículo
en Inglés
| MEDLINE | ID: mdl-32512884
18.
Limitations in a frataxin knockdown cell model for Friedreich ataxia in a high-throughput drug screen.
BMC Neurol
; 9: 46, 2009 Aug 24.
Artículo
en Inglés
| MEDLINE | ID: mdl-19703283
19.
Hypoxic Environment and Paired Hierarchical 3D and 2D Models of Pediatric H3.3-Mutated Gliomas Recreate the Patient Tumor Complexity.
Cancers (Basel)
; 11(12)2019 Nov 26.
Artículo
en Inglés
| MEDLINE | ID: mdl-31779235
20.
SynAggreg: A Multifunctional High-Throughput Technology for Precision Study of Amyloid Aggregation and Systematic Discovery of Synergistic Inhibitor Compounds.
J Mol Biol
; 430(24): 5257-5279, 2018 12 07.
Artículo
en Inglés
| MEDLINE | ID: mdl-30266595