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1.
Tranylcypromine-Based LSD1 Inhibitors: Structure-Activity Relationships, Antiproliferative Effects in Leukemia, and Gene Target Modulation.
ChemMedChem
; 15(7): 643-658, 2020 04 03.
Artículo
en Inglés
| MEDLINE | ID: mdl-32003940
2.
Discovery of Reversible Inhibitors of KDM1A Efficacious in Acute Myeloid Leukemia Models.
ACS Med Chem Lett
; 11(5): 754-759, 2020 May 14.
Artículo
en Inglés
| MEDLINE | ID: mdl-32435381
3.
New 6- and 7-heterocyclyl-1H-indole derivatives as potent tubulin assembly and cancer cell growth inhibitors.
Eur J Med Chem
; 152: 283-297, 2018 May 25.
Artículo
en Inglés
| MEDLINE | ID: mdl-29730191
4.
Thieno[3,2-b]pyrrole-5-carboxamides as New Reversible Inhibitors of Histone Lysine Demethylase KDM1A/LSD1. Part 2: Structure-Based Drug Design and Structure-Activity Relationship.
J Med Chem
; 60(5): 1693-1715, 2017 03 09.
Artículo
en Inglés
| MEDLINE | ID: mdl-28186757
5.
3-Aroyl-1,4-diarylpyrroles Inhibit Chronic Myeloid Leukemia Cell Growth through an Interaction with Tubulin.
ACS Med Chem Lett
; 8(5): 521-526, 2017 May 11.
Artículo
en Inglés
| MEDLINE | ID: mdl-28523104
6.
Thieno[3,2-b]pyrrole-5-carboxamides as New Reversible Inhibitors of Histone Lysine Demethylase KDM1A/LSD1. Part 1: High-Throughput Screening and Preliminary Exploration.
J Med Chem
; 60(5): 1673-1692, 2017 03 09.
Artículo
en Inglés
| MEDLINE | ID: mdl-28186755
7.
Effect of tamoxifen in an experimental model of breast tumor studied by dynamic contrast-enhanced magnetic resonance imaging and different contrast agents.
Invest Radiol
; 40(7): 421-9, 2005 Jul.
Artículo
en Inglés
| MEDLINE | ID: mdl-15973133
8.
New Indole Tubulin Assembly Inhibitors Cause Stable Arrest of Mitotic Progression, Enhanced Stimulation of Natural Killer Cell Cytotoxic Activity, and Repression of Hedgehog-Dependent Cancer.
J Med Chem
; 58(15): 5789-807, 2015 Aug 13.
Artículo
en Inglés
| MEDLINE | ID: mdl-26132075
9.
Chiral resolution and pharmacological characterization of the enantiomers of the Hsp90 inhibitor 2-amino-7-[4-fluoro-2-(3-pyridyl)phenyl]-4-methyl-7,8-dihydro-6H-quinazolin-5-one oxime.
ChemMedChem
; 9(7): 1574-85, 2014 Jul.
Artículo
en Inglés
| MEDLINE | ID: mdl-24753447
10.
New pyrrole derivatives with potent tubulin polymerization inhibiting activity as anticancer agents including hedgehog-dependent cancer.
J Med Chem
; 57(15): 6531-52, 2014 Aug 14.
Artículo
en Inglés
| MEDLINE | ID: mdl-25025991
11.
Synthesis and biological characterization of spiro[2H-(1,3)-benzoxazine-2,4'-piperidine] based histone deacetylase inhibitors.
Eur J Med Chem
; 64: 273-84, 2013 Jun.
Artículo
en Inglés
| MEDLINE | ID: mdl-23644210
12.
Toward highly potent cancer agents by modulating the C-2 group of the arylthioindole class of tubulin polymerization inhibitors.
J Med Chem
; 56(1): 123-49, 2013 Jan 10.
Artículo
en Inglés
| MEDLINE | ID: mdl-23214452
13.
Spiro[chromane-2,4'-piperidine]-based histone deacetylase inhibitors with improved in vivo activity.
ChemMedChem
; 7(4): 709-21, 2012 Apr.
Artículo
en Inglés
| MEDLINE | ID: mdl-22354629
14.
Synthesis and biological evaluation of N-hydroxyphenylacrylamides and N-hydroxypyridin-2-ylacrylamides as novel histone deacetylase inhibitors.
J Med Chem
; 53(2): 822-39, 2010 Jan 28.
Artículo
en Inglés
| MEDLINE | ID: mdl-20017493
15.
Contrast-enhanced MRI of murine sponge model for progressive angiogenesis assessed with gadoteridol (ProHance) and gadocoletic acid trisodium salt (B22956/1).
J Magn Reson Imaging
; 27(4): 872-80, 2008 Apr.
Artículo
en Inglés
| MEDLINE | ID: mdl-18383249
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