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1.
Scaffold oriented synthesis. Part 4: design, synthesis and biological evaluation of novel 5-substituted indazoles as potent and selective kinase inhibitors employing heterocycle forming and multicomponent reactions.
Bioorg Med Chem Lett
; 21(5): 1480-3, 2011 Mar 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-21288717
2.
Scaffold oriented synthesis. Part 3: design, synthesis and biological evaluation of novel 5-substituted indazoles as potent and selective kinase inhibitors employing [2+3] cycloadditions.
Bioorg Med Chem Lett
; 21(5): 1476-9, 2011 Mar 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-21282054
3.
Structure-Based Design of A-1293102, a Potent and Selective BCL-XL Inhibitor.
ACS Med Chem Lett
; 12(6): 1011-1016, 2021 Jun 10.
Artículo
en Inglés
| MEDLINE | ID: mdl-34141086
4.
Bacterial translation inhibitors, 1-acylindazol-3-ols as anthranilic acid mimics.
Bioorg Med Chem Lett
; 18(23): 6293-7, 2008 Dec 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-18951783
5.
cis-4-(Piperazin-1-yl)-5,6,7a,8,9,10,11,11a-octahydrobenzofuro[2,3-h]quinazolin-2-amine (A-987306), a new histamine H4R antagonist that blocks pain responses against carrageenan-induced hyperalgesia.
J Med Chem
; 51(22): 7094-8, 2008 Nov 27.
Artículo
en Inglés
| MEDLINE | ID: mdl-18983139
6.
Preparation of novel anthranilic acids as antibacterial agents: extensive evaluation of structural and physical properties on antibacterial activity and human serum albumin affinity.
Bioorg Med Chem Lett
; 17(11): 3113-6, 2007 Jun 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-17400450
7.
Structure-activity relationships of bioisosteres of a carboxylic acid in a novel class of bacterial translation inhibitors.
Bioorg Med Chem Lett
; 17(14): 4040-3, 2007 Jul 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-17561394
8.
Preparation of novel antibacterial agents. Replacement of the central aromatic ring with heterocycles.
Bioorg Med Chem Lett
; 17(8): 2347-50, 2007 Apr 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-17350254
9.
Preparation of novel anthranilic acids as antibacterial agents. Extensive evaluation of alternative amide bioisosteres connecting the A- and the B-rings.
Bioorg Med Chem Lett
; 17(10): 2823-7, 2007 May 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-17368020
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