Detalles de la búsqueda
1.
A New Paroxetine-Based GRK2 Inhibitor Reduces Internalization of the µ-Opioid Receptor.
Mol Pharmacol
; 97(6): 392-401, 2020 06.
Artículo
en Inglés
| MEDLINE | ID: mdl-32234810
2.
Small-Molecule G Protein-Coupled Receptor Kinase Inhibitors Attenuate G Protein-Coupled Receptor Kinase 2-Mediated Desensitization of Vasoconstrictor-Induced Arterial Contractions.
Mol Pharmacol
; 94(3): 1079-1091, 2018 09.
Artículo
en Inglés
| MEDLINE | ID: mdl-29980659
3.
Utilizing a structure-based docking approach to develop potent G protein-coupled receptor kinase (GRK) 2 and 5 inhibitors.
Bioorg Med Chem Lett
; 28(9): 1507-1515, 2018 05 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-29627263
4.
Structural Determinants Influencing the Potency and Selectivity of Indazole-Paroxetine Hybrid G Protein-Coupled Receptor Kinase 2 Inhibitors.
Mol Pharmacol
; 92(6): 707-717, 2017 12.
Artículo
en Inglés
| MEDLINE | ID: mdl-29070696
5.
Crystal Structure of G Protein-coupled Receptor Kinase 5 in Complex with a Rationally Designed Inhibitor.
J Biol Chem
; 290(34): 20649-20659, 2015 Aug 21.
Artículo
en Inglés
| MEDLINE | ID: mdl-26032411
6.
Translation of structure-activity relationships from cyclic mixed efficacy opioid peptides to linear analogues.
Biopolymers
; 102(1): 107-14, 2014 Jan.
Artículo
en Inglés
| MEDLINE | ID: mdl-24436042
7.
Structure-Based Design of Selective, Covalent G Protein-Coupled Receptor Kinase 5 Inhibitors.
ACS Med Chem Lett
; 10(12): 1628-1634, 2019 Dec 12.
Artículo
en Inglés
| MEDLINE | ID: mdl-31857838
8.
Structure-Based Design of Highly Selective and Potent G Protein-Coupled Receptor Kinase 2 Inhibitors Based on Paroxetine.
J Med Chem
; 60(7): 3052-3069, 2017 04 13.
Artículo
en Inglés
| MEDLINE | ID: mdl-28323425
9.
Occludin S471 Phosphorylation Contributes to Epithelial Monolayer Maturation.
Mol Cell Biol
; 36(15): 2051-66, 2016 08 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-27185880
10.
Structure-Based Design, Synthesis, and Biological Evaluation of Highly Selective and Potent G Protein-Coupled Receptor Kinase 2 Inhibitors.
J Med Chem
; 59(8): 3793-807, 2016 04 28.
Artículo
en Inglés
| MEDLINE | ID: mdl-27050625
11.
Correction to "Structure-Based Design of Highly Selective and Potent G Protein-Coupled Receptor Kinase 2 Inhibitors Based on Paroxetine".
J Med Chem
; 62(12): 5920, 2019 Jun 27.
Artículo
en Inglés
| MEDLINE | ID: mdl-31188593
Resultados
1 -
11
de 11
1
Próxima >
>>