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1.
Multifaceted roles for BCL3 in cancer: a proto-oncogene comes of age.
Mol Cancer
; 23(1): 7, 2024 01 09.
Artículo
en Inglés
| MEDLINE | ID: mdl-38195591
2.
Design, Synthesis, and Potent Anticancer Activity of Novel Indole-Based Bcl-2 Inhibitors.
Int J Mol Sci
; 24(19)2023 Sep 28.
Artículo
en Inglés
| MEDLINE | ID: mdl-37834104
3.
Whole blood-based measurement of SARS-CoV-2-specific T cells reveals asymptomatic infection and vaccine immunogenicity in healthy subjects and patients with solid-organ cancers.
Immunology
; 165(2): 250-259, 2022 02.
Artículo
en Inglés
| MEDLINE | ID: mdl-34775604
4.
Synthesis, biological evaluation and X-ray analysis of bicalutamide sulfoxide analogues for the potential treatment of prostate cancer.
Bioorg Med Chem Lett
; 36: 127817, 2021 03 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-33513386
5.
New Bioactive Fused Triazolothiadiazoles as Bcl-2-Targeted Anticancer Agents.
Int J Mol Sci
; 22(22)2021 Nov 12.
Artículo
en Inglés
| MEDLINE | ID: mdl-34830153
6.
Design, Synthesis and Evaluation of New Bioactive Oxadiazole Derivatives as Anticancer Agents Targeting Bcl-2.
Int J Mol Sci
; 21(23)2020 Nov 26.
Artículo
en Inglés
| MEDLINE | ID: mdl-33256166
7.
Synthesis and Biological Evaluation of Bicalutamide Analogues for the Potential Treatment of Prostate Cancer.
Molecules
; 26(1)2020 Dec 24.
Artículo
en Inglés
| MEDLINE | ID: mdl-33374450
8.
Structure-Based Virtual Screening, Synthesis and Biological Evaluation of Potential FAK-FAT Domain Inhibitors for Treatment of Metastatic Cancer.
Molecules
; 25(15)2020 Jul 31.
Artículo
en Inglés
| MEDLINE | ID: mdl-32751931
9.
Radiosynthesis of [18F]-Labelled Pro-Nucleotides (ProTides).
Molecules
; 25(3)2020 Feb 06.
Artículo
en Inglés
| MEDLINE | ID: mdl-32041321
10.
Polyfluoroaromatic stavudine (d4T) ProTides exhibit enhanced anti-HIV activity.
Bioorg Med Chem Lett
; 29(24): 126721, 2019 12 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-31679972
11.
New Quinoline-Based Heterocycles as Anticancer Agents Targeting Bcl-2.
Molecules
; 24(7)2019 Apr 02.
Artículo
en Inglés
| MEDLINE | ID: mdl-30986908
12.
Pharmacologically directed strategies in academic anticancer drug discovery based on the European NCI compounds initiative.
Br J Cancer
; 117(2): 195-202, 2017 Jul 11.
Artículo
en Inglés
| MEDLINE | ID: mdl-28609434
13.
Synthesis and evaluation of 5-(1H-indol-3-yl)-N-aryl-1,3,4-oxadiazol-2-amines as Bcl-2 inhibitory anticancer agents.
Bioorg Med Chem Lett
; 27(4): 1037-1040, 2017 02 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-28087272
14.
7-Substituted umbelliferone derivatives as androgen receptor antagonists for the potential treatment of prostate and breast cancer.
Bioorg Med Chem Lett
; 26(8): 2000-4, 2016 Apr 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-26965862
15.
Synthesis and in vitro anticancer evaluation of some 4,6-diamino-1,3,5-triazine-2-carbohydrazides as Rad6 ubiquitin conjugating enzyme inhibitors.
Bioorg Med Chem Lett
; 26(8): 2030-4, 2016 Apr 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-26965855
16.
ProTides of BVdU as potential anticancer agents upon efficient intracellular delivery of their activated metabolites.
Bioorg Med Chem Lett
; 26(23): 5618-5623, 2016 12 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-27818111
17.
Rational design and synthesis of novel anti-prostate cancer agents bearing a 3,5-bis-trifluoromethylphenyl moiety.
Bioorg Med Chem Lett
; 26(15): 3636-40, 2016 08 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-27301368
18.
Novel indole-based melatonin analogues substituted with triazole, thiadiazole and carbothioamides: studies on their antioxidant, chemopreventive and cytotoxic activities.
J Enzyme Inhib Med Chem
; 31(6): 1312-21, 2016 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-26745200
19.
Gold nanoparticle conjugated Rad6 inhibitor induces cell death in triple negative breast cancer cells by inducing mitochondrial dysfunction and PARP-1 hyperactivation: Synthesis and characterization.
Nanomedicine
; 12(3): 745-757, 2016 Apr.
Artículo
en Inglés
| MEDLINE | ID: mdl-26563438
20.
Synthesis, anti-HIV and cytostatic evaluation of 3'-deoxy-3'-fluorothymidine (FLT) pro-nucleotides.
Bioorg Med Chem Lett
; 24(10): 2240-3, 2014 May 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-24751439