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1.
Discovery of novel BRD4 inhibitors by high-throughput screening, crystallography, and cell-based assays.
Bioorg Med Chem Lett
; 27(9): 2003-2009, 2017 05 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-28347667
2.
Discovery of novel BET inhibitors by drug repurposing of nitroxoline and its analogues.
Org Biomol Chem
; 15(44): 9352-9361, 2017 Nov 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-29087414
3.
Machine-Learning-Assisted Approach for Discovering Novel Inhibitors Targeting Bromodomain-Containing Protein 4.
J Chem Inf Model
; 57(7): 1677-1690, 2017 07 24.
Artículo
en Inglés
| MEDLINE | ID: mdl-28636361
4.
Molecular Mechanism underlying PRMT1 Dimerization for SAM Binding and Methylase Activity.
J Chem Inf Model
; 55(12): 2623-32, 2015 Dec 28.
Artículo
en Inglés
| MEDLINE | ID: mdl-26562720
5.
Discovery of two aminoglycoside antibiotics as inhibitors targeting the menin-mixed lineage leukaemia interface.
Bioorg Med Chem Lett
; 24(9): 2090-3, 2014 May 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-24709560
6.
Virtual screening and biological evaluation of novel small molecular inhibitors against protein arginine methyltransferase 1 (PRMT1).
Org Biomol Chem
; 12(47): 9665-73, 2014 Dec 21.
Artículo
en Inglés
| MEDLINE | ID: mdl-25348815
7.
pH-responsive pickering foam created from self-aggregate polymer using dynamic covalent bond.
J Colloid Interface Sci
; 597: 383-392, 2021 Sep.
Artículo
en Inglés
| MEDLINE | ID: mdl-33894546
8.
PRMT1 is a novel molecular therapeutic target for clear cell renal cell carcinoma.
Theranostics
; 11(11): 5387-5403, 2021.
Artículo
en Inglés
| MEDLINE | ID: mdl-33859753
9.
Discovery of trisubstituted nicotinonitrile derivatives as novel human GCN5 inhibitors through AlphaScreen-based high throughput screening.
RSC Adv
; 9(9): 4917-4924, 2019 Feb 05.
Artículo
en Inglés
| MEDLINE | ID: mdl-35514635
10.
Development and evaluation of a novel series of Nitroxoline-derived BET inhibitors with antitumor activity in renal cell carcinoma.
Oncogenesis
; 7(11): 83, 2018 Nov 02.
Artículo
en Inglés
| MEDLINE | ID: mdl-30385738
11.
Development of Potent Type I Protein Arginine Methyltransferase (PRMT) Inhibitors of Leukemia Cell Proliferation.
J Med Chem
; 60(21): 8888-8905, 2017 11 09.
Artículo
en Inglés
| MEDLINE | ID: mdl-29019697
12.
Discovery of novel trimethoxy-ring BRD4 bromodomain inhibitors: AlphaScreen assay, crystallography and cell-based assay.
Medchemcomm
; 8(6): 1322-1331, 2017 Jun 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-30108844
13.
Discovery of alkyl bis(oxy)dibenzimidamide derivatives as novel protein arginine methyltransferase 1 (PRMT1) inhibitors.
Chem Biol Drug Des
; 90(6): 1260-1270, 2017 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-28636189
14.
Identification of Novel Inhibitors against Coactivator Associated Arginine Methyltransferase 1 Based on Virtual Screening and Biological Assays.
Biomed Res Int
; 2016: 7086390, 2016.
Artículo
en Inglés
| MEDLINE | ID: mdl-27872854
15.
Discovery and Optimization of Novel, Selective Histone Methyltransferase SET7 Inhibitors by Pharmacophore- and Docking-Based Virtual Screening.
J Med Chem
; 58(20): 8166-81, 2015 Oct 22.
Artículo
en Inglés
| MEDLINE | ID: mdl-26390175
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