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1.
Structure-based linker exploration: Discovery of 1-ethyl-1H-indole analogs as novel ATX inhibitors.
Bioorg Med Chem
; 28(22): 115795, 2020 11 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-33032188
2.
Design, synthesis and biological evaluation of 2-arylaminopyrimidine derivatives bearing 1,3,8-triazaspiro[4,5]decan-4-one or piperidine-3-carboxamide moiety as novel Type-I1/2 ALK inhibitors.
Bioorg Chem
; 94: 103456, 2020 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-31787343
3.
Discovery and optimization of tetrahydropyrido[4,3-d]pyrimidine derivatives as novel ATX and EGFR dual inhibitors.
Bioorg Med Chem
; 26(8): 1784-1796, 2018 05 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-29496411
4.
Design, synthesis and biological evaluation N2-(2-alkyoxy-6-aliphatic aminopyridin-3-yl)-2,4-diaminepyrimidine derivatives bearing acylamino or DBTD 'head' as potential ALK inhibitors.
Bioorg Chem
; 81: 689-699, 2018 12.
Artículo
en Inglés
| MEDLINE | ID: mdl-30268049
5.
Synthesis, biological evaluation and molecular modeling of imidazo[1,2-a]pyridine derivatives as potent antitubulin agents.
Bioorg Med Chem
; 25(15): 4088-4099, 2017 08 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-28622907
6.
Discovery of novel mutant-combating ALK and ROS1 dual inhibitors bearing imidazolidin-2-one moiety with reasonable PK properties.
Eur J Med Chem
; 171: 297-309, 2019 Jun 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-30927566
7.
Dual potent ALK and ROS1 inhibitors combating drug-resistant mutants: Synthesis and biological evaluation of aminopyridine-containing diarylaminopyrimidine derivatives.
Eur J Med Chem
; 158: 322-333, 2018 Oct 05.
Artículo
en Inglés
| MEDLINE | ID: mdl-30223120
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