Detalles de la búsqueda
1.
Identification of 1-Methyl-N-(propan-2-yl)-N-({2-[4-(trifluoromethoxy)phenyl]pyridin-4-yl}methyl)-1H-imidazole-4-carboxamide as a Potent and Orally Available Glycine Transporter 1 Inhibitor.
Chem Pharm Bull (Tokyo)
; 64(11): 1630-1640, 2016.
Artículo
en Inglés
| MEDLINE | ID: mdl-27803474
2.
Antipsychotic profiles of TASP0443294, a novel and orally active positive allosteric modulator of metabotropic glutamate 2 receptor.
J Pharmacol Sci
; 127(3): 352-61, 2015 Mar.
Artículo
en Inglés
| MEDLINE | ID: mdl-25837934
3.
Neurophysiologic and antipsychotic profiles of TASP0433864, a novel positive allosteric modulator of metabotropic glutamate 2 receptor.
J Pharmacol Exp Ther
; 351(3): 642-53, 2014 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-25277141
4.
Synthesis, in vitro pharmacology, and pharmacokinetic profiles of 2-[1-amino-1-carboxy-2-(9H-xanthen-9-yl)-ethyl]-1-fluorocyclopropanecarboxylic acid and its 6-heptyl ester, a potent mGluR2 antagonist.
Bioorg Med Chem
; 16(8): 4359-66, 2008 Apr 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-18348906
5.
Neuropharmacological profiles of antagonists of group II metabotropic glutamate receptors.
Neurosci Lett
; 378(3): 131-4, 2005 Apr 22.
Artículo
en Inglés
| MEDLINE | ID: mdl-15781145
6.
MGS0039: a potent and selective group II metabotropic glutamate receptor antagonist with antidepressant-like activity.
Neuropharmacology
; 46(4): 457-67, 2004 Mar.
Artículo
en Inglés
| MEDLINE | ID: mdl-14975669
7.
Synthesis, in vitro pharmacology, structure-activity relationships, and pharmacokinetics of 3-alkoxy-2-amino-6-fluorobicyclo[3.1.0]hexane-2,6-dicarboxylic acid derivatives as potent and selective group II metabotropic glutamate receptor antagonists.
J Med Chem
; 47(18): 4570-87, 2004 Aug 26.
Artículo
en Inglés
| MEDLINE | ID: mdl-15317467
8.
Metabotropic glutamate receptors: potential drug targets for psychiatric disorders.
Open Med Chem J
; 4: 20-36, 2010 May 27.
Artículo
en Inglés
| MEDLINE | ID: mdl-21160908
9.
In vitro and in vivo evaluation of the metabolism and bioavailability of ester prodrugs of mgs0039 (3-(3,4-dichlorobenzyloxy)-2-amino-6-fluorobicyclo[3.1.0]hexane-2,6-dicarboxylic Acid), a potent metabotropic glutamate receptor antagonist.
Drug Metab Dispos
; 34(3): 369-74, 2006 Mar.
Artículo
en Inglés
| MEDLINE | ID: mdl-16326817
10.
Synthesis, in vitro pharmacology, and structure-activity relationships of 2-aminobicyclo[3.1.0]hexane-2,6-dicarboxylic acid derivatives as mGluR2 antagonists.
Bioorg Med Chem
; 14(10): 3405-20, 2006 May 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-16431115
11.
Prodrugs of 3-(3,4-dichlorobenzyloxy)-2-amino-6-fluorobicyclo[3.1.0]hexane-2,6-dicarboxylic acid (MGS0039): a potent and orally active group II mGluR antagonist with antidepressant-like potential.
Bioorg Med Chem
; 14(12): 4193-207, 2006 Jun 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-16487713
12.
A concise synthesis of furostifoline by tetrabutylammonium fluoride-promoted indole ring formation.
Chem Pharm Bull (Tokyo)
; 50(1): 143-5, 2002 Jan.
Artículo
en Inglés
| MEDLINE | ID: mdl-11824578
13.
Convenient indole synthesis from 2-iodoanilines and terminal alkynes by the sequential Sonogashira reaction and the cyclization reaction promoted by tetrabutylammonium fluoride (TBAF).
Chem Pharm Bull (Tokyo)
; 51(10): 1170-3, 2003 Oct.
Artículo
en Inglés
| MEDLINE | ID: mdl-14519923
14.
Synthesis of 2,3-disubstituted indole using palladium(II)-catalyzed cyclization with alkenylation reaction.
Chem Pharm Bull (Tokyo)
; 50(2): 235-8, 2002 Feb.
Artículo
en Inglés
| MEDLINE | ID: mdl-11848216
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