1.
Org Lett
; 14(9): 2202-5, 2012 May 04.
Article
in English
| MEDLINE
| ID: mdl-22506630
ABSTRACT
A novel approach for the direct C-4 arylation of N-methyl-1,2,3,4-tetrahydroisoquinolines by nucleophilic addition of ß-aminocarbanions to benzynes is described which provides a one-pot procedure for synthesis of the title compounds.