1.
Amino Acids
; 48(9): 2237-42, 2016 09.
Article
in English
| MEDLINE
| ID: mdl-27206723
ABSTRACT
We synthesized in a few steps both diastereomers of orthogonally protected ß,γ-diamino acids starting from L-phenylalanine or L-tryptophan. These final compounds are interesting building blocks for peptide synthesis and foldamer chemistry. The key step is a Blaise reaction performed under ultrasound conditions.
Subject(s)
Phenylalanine/chemistry , Phenylalanine/chemical synthesis , Tryptophan/chemistry , Tryptophan/chemical synthesis , Ultrasonic Waves , Stereoisomerism
2.
Bioorg Med Chem Lett
; 14(12): 3303-6, 2004 Jun 21.
Article
in English
| MEDLINE
| ID: mdl-15149695
Subject(s)
3',5'-Cyclic-AMP Phosphodiesterases/antagonists & inhibitors , Cycloheptanes/chemistry , Phosphodiesterase Inhibitors/chemistry , 3',5'-Cyclic-AMP Phosphodiesterases/metabolism , Azulenes , Cyclic Nucleotide Phosphodiesterases, Type 4 , Cycloheptanes/pharmacology , Phosphodiesterase Inhibitors/pharmacology
3.
Angew Chem Int Ed Engl
; 41(6): 979-82, 2002 Mar 15.
Article
in English
| MEDLINE
| ID: mdl-12491287