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Bioorg Med Chem Lett
; 15(1): 93-8, 2005 Jan 03.
Article
in English
| MEDLINE
| ID: mdl-15582418
ABSTRACT
A series of non-amide-linked 6-substituted-2-naphthamidine urokinase plasminogen activator (uPA) inhibitors are described. These compounds possess excellent binding activities and selectivities with significantly improved pharmacokinetic profiles versus previously described amide-linked inhibitors.
