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Bioorg Med Chem Lett
; 23(15): 4370-3, 2013 Aug 01.
Article
in English
| MEDLINE
| ID: mdl-23777782
ABSTRACT
A series of potent α4ß1/α4ß7 integrin inhibitors is reported, including an inhibitor 12d with remarkable oral exposure and efficacy in rat models of rheumatoid arthritis and Crohn's disease.