1.
Bioorg Med Chem Lett
; 13(7): 1291-2, 2003 Apr 07.
Article
in English
| MEDLINE
| ID: mdl-12657266
ABSTRACT
The synthesis of NPTS, 6, a potent inhibitor of the type 1 glycine transporter (GlyT1) is described, as well as preparation of 6 in optically active and tritiated form for use as a radioligand for affinity displacement assay of GlyT1.