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Bioorg Med Chem Lett
; 16(23): 6086-90, 2006 Dec 01.
Article
in English
| MEDLINE
| ID: mdl-16987661
ABSTRACT
A series of potent steroidal glucocorticoid receptor antagonists has been discovered. After conjugation to cholic acid, the compounds retained an affinity for GR in vitro and had modest in vivo efficacy.