1.
Chem Commun (Camb)
; 55(7): 929-932, 2019 Jan 17.
Article
in English
| MEDLINE
| ID: mdl-30601480
ABSTRACT
A preloaded resin consisting of a thalidomide moiety and an ethylene-oxy linker allows the simple and fast formation of PROTACs. The feasibility of the procedure was illustrated by conjugating different protein kinase inhibitors. The biological functionality of an ibrutinib-like conjugate was then confirmed by a cellular experiment.
2.
Vnitr Lek
; 27(10): 948-56, 1981 Oct.
Article
in Slovak
| MEDLINE
| ID: mdl-7314534