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Novel benzopyrano[3,4-c]pyrrole derivatives as potent and selective dopamine D3 receptor antagonist.
Bioorg Med Chem Lett
; 9(14): 2059-64, 1999 Jul 19.
Article
in English
| MEDLINE
| ID: mdl-10450981
ABSTRACT
A new series of benzopyrano[3,4-c]pyrrole derivatives were synthesized and evaluated for their interaction with dopamine D3 versus D2 receptors. Amongst these compounds, 4x (S 33084) was found to be a potent and selective dopamine D3 receptor antagonist.