1.
Bioorg Med Chem Lett
; 17(11): 3109-12, 2007 Jun 01.
Article
in English
| MEDLINE
| ID: mdl-17383873
ABSTRACT
The synthesis, biological activity, and pharmacokinetic profile of CCR1 antagonists are described.
Subject(s)
Piperazines/chemistry , Piperazines/metabolism , Receptors, Chemokine/antagonists & inhibitors , Animals , Dogs , Haplorhini , Humans , Microsomes, Liver/metabolism , Piperazines/chemical synthesis , Rats , Receptors, CCR1
2.
Bioorg Med Chem Lett
; 14(9): 2175-9, 2004 May 03.
Article
in English
| MEDLINE
| ID: mdl-15081003
ABSTRACT
The synthesis, biological activity, and pharmacokinetic profile of novel CCR1 antagonists are described.