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Bioorg Med Chem Lett
; 29(14): 1746-1748, 2019 07 15.
Article
in English
| MEDLINE
| ID: mdl-31103445
ABSTRACT
Structure based virtual screening attempts to discover DUSP1 inhibitors have yielded a scaffold featuring benzoxazole and acylthiourea pharmacophore. A series of its analogues were synthesized to explore structure activity relationship (SAR) of DUSP1 inhibition.