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2.
Indian J Physiol Pharmacol ; 25(3): 269-73, 1981.
Article in English | MEDLINE | ID: mdl-7298153

ABSTRACT

Benzamido (alkyl) methyl pyrrolidine Mannich bases were synthetized and subjected to certain neuropharmacological studies. All the bases reduced the pentobarbitone sleeping time and rota-rod grip of rats. The Mannich bases II, III and V raised the minimal electro-shock seizure threshold of rats. The TAB-induced pyrexia was not reduced by the bases I and III in rabbits. None of the bases showed any significant analgesic activity.


Subject(s)
Amines/pharmacology , Brain/drug effects , Mannich Bases/pharmacology , Receptors, Drug/metabolism , Animals , Body Temperature/drug effects , Brain/metabolism , Male , Pentobarbital/pharmacology , Postural Balance/drug effects , Rabbits , Rats , Sensory Thresholds/drug effects , Sleep/drug effects , Time Factors
5.
Indian J Physiol Pharmacol ; 20(3): 168-71, 1976.
Article in English | MEDLINE | ID: mdl-977086

ABSTRACT

Intraventricular injection of histamine and normal saline in rats caused a marked fall in adrenal ascorbic acid indicating a stimulatory effect of both on pituitary adrenal axis. Intraventricularly injected histamine caused significant hypoglycaemia also in rats as compared to control series.


Subject(s)
Adrenal Glands/drug effects , Blood Glucose/analysis , Histamine/pharmacology , Hypothalamus/drug effects , Pituitary Gland/drug effects , Adrenal Glands/analysis , Animals , Ascorbic Acid/analysis , Depression, Chemical , Histamine/administration & dosage , Injections, Intraventricular , Rats
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