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Bioorg Med Chem Lett
; 12(3): 315-8, 2002 Feb 11.
Article
in English
| MEDLINE
| ID: mdl-11814786
ABSTRACT
Fluorescent analogues of the cholesterol absorption inhibitor (CAI), Sch 58235, have been designed and synthesized as single enantiomers. Biological testing reveals that they are potent CAIs and are suitable tools for the investigation of the azetidinone CAI mechanism of action (MOA).