1.
Bioorg Med Chem Lett
; 17(1): 73-7, 2007 Jan 01.
Artículo
en Inglés
| MEDLINE
| ID: mdl-17046251
RESUMEN
We describe a novel series of potent inhibitors of human beta-secretase. These compounds possess the hydroxyethyl amine transition state isostere. A 2.5A crystal structure of inhibitor 32 bound to BACE is provided.