1.
J Org Chem
; 81(1): 256-64, 2016 Jan 04.
Artigo
em Inglês
| MEDLINE
| ID: mdl-26624806
RESUMO
Intramolecular Pd-catalyzed functionalization of cyclopropyl α-amino acid-derived benzamides proceeds without silver or pivalate additives. Both electronically and sterically diverse ethyl 1,2,3,4-tetrahydroisoquinolone-3-carboxylates were accessible in good to excellent yields.