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Bull Exp Biol Med ; 134(1): 8-11, 2002 Jul.
Artigo em Inglês | MEDLINE | ID: mdl-12459855

RESUMO

The effect of 5-hydroxytryptamine (serotonin) on neuromuscular transmission in frog skeletal muscle was studied using voltage clamp technique. Serotonin produced no effect on end-plate currents during low frequency electrical stimulation of the motor nerve, but increased the amplitude depression of multiquantal currents during high-frequency stimulation similar to motor commands fired by motoneurons. It was shown that the inhibitory effect of serotonin on neuromuscular transmission is determined by slow potential-dependent block of open ionic channels in the postsynaptic membrane accumulating during rhythmic activation of the synapse.


Assuntos
Músculo Esquelético/efeitos dos fármacos , Serotonina/farmacologia , Acetilcolina/metabolismo , Acetilcolinesterase/farmacologia , Animais , Eletrofisiologia , Íons , Potenciais da Membrana , Músculo Esquelético/metabolismo , Neostigmina/farmacologia , Neurônios/metabolismo , Ranidae , Nervo Isquiático/metabolismo , Serotonina/metabolismo , Fatores de Tempo
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