1.
Gen Pharmacol
; 30(4): 521-4, 1998 Apr.
Artigo
em Inglês
| MEDLINE
| ID: mdl-9522169
RESUMO
1. A study has been made to know the effects of clozapine and clothiapine on the responses of rat isolated vas deferens to norepinephrine, dopamine and potassium, those of the rat isolated uterus to serotonin and potassium, and that of guinea pig isolated ileum to histamine. 2. Clozapine was a noncompetitive antagonist to norepinephrine, dopamine, serotonin and histamine; it inhibited potassium-induced contraction in isolated rat uterus and vas deferens. 3. Clothiapine was a competitive antagonist to serotonin and a noncompetitive antagonist to norepinephrine, dopamine and histamine; it inhibited potassium-induced contractions in isolated rat uterus and vas deferens.
Assuntos
Antipsicóticos/farmacologia , Clozapina/farmacologia , Dibenzotiazepinas/farmacologia , Íleo/efeitos dos fármacos , Contração Muscular/efeitos dos fármacos , Útero/efeitos dos fármacos , Ducto Deferente/efeitos dos fármacos , Animais , Relação Dose-Resposta a Droga , Feminino , Cobaias , Íleo/fisiologia , Masculino , Ratos , Ratos Wistar , Útero/fisiologia
2.
Rev Clin Esp
; 189(8): 391-2, 1991 Nov.
Artigo
em Espanhol
| MEDLINE
| ID: mdl-1784806