1.
J Org Chem
; 88(19): 13686-13698, 2023 Oct 06.
Artigo
em Inglês
| MEDLINE
| ID: mdl-37767971
RESUMO
We have described a dual palladium-photoredox-catalyzed highly regioselective acylation of carbazoles and indolines using molecular oxygen as the green oxidant. The reaction shows a broad substrate scope and good functional group tolerance. Late-stage functionalization of a carprofen drug derivative, further manipulation of products, and gram-scale synthesis of the acylated products were illustrated to show the versatility of the method.