1.
Bioorg Med Chem Lett
; 12(24): 3565-7, 2002 Dec 16.
Artigo
em Inglês
| MEDLINE
| ID: mdl-12443777
RESUMO
A series of 5-substituted 2-benzoylaminobenzoic acids has been synthesized and assayed for PPARalpha/gamma activity. Both dual activators and selective PPARgamma agonists have been identified. This class of compounds was shown to activate the PPARgamma receptor through interaction with a novel binding site.