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Potent and Selective CK2 Kinase Inhibitors with Effects on Wnt Pathway Signaling in Vivo.
Dowling, James E; Alimzhanov, Marat; Bao, Larry; Chuaqui, Claudio; Denz, Christopher R; Jenkins, Emma; Larsen, Nicholas A; Lyne, Paul D; Pontz, Timothy; Ye, Qing; Holdgate, Geoff A; Snow, Lindsay; O'Connell, Nichole; Ferguson, Andrew D.
Affiliation
  • Dowling JE; Oncology Innovative Medicines Unit, AstraZeneca R&D , 35 Gatehouse Drive, Waltham, Massachusetts 02451, United States.
  • Alimzhanov M; Oncology Innovative Medicines Unit, AstraZeneca R&D , 35 Gatehouse Drive, Waltham, Massachusetts 02451, United States.
  • Bao L; Oncology Innovative Medicines Unit, AstraZeneca R&D , 35 Gatehouse Drive, Waltham, Massachusetts 02451, United States.
  • Chuaqui C; Oncology Innovative Medicines Unit, AstraZeneca R&D , 35 Gatehouse Drive, Waltham, Massachusetts 02451, United States.
  • Denz CR; Oncology Innovative Medicines Unit, AstraZeneca R&D , 35 Gatehouse Drive, Waltham, Massachusetts 02451, United States.
  • Jenkins E; Oncology Innovative Medicines Unit, AstraZeneca R&D , 35 Gatehouse Drive, Waltham, Massachusetts 02451, United States.
  • Larsen NA; Oncology Innovative Medicines Unit, AstraZeneca R&D , 35 Gatehouse Drive, Waltham, Massachusetts 02451, United States.
  • Lyne PD; Oncology Innovative Medicines Unit, AstraZeneca R&D , 35 Gatehouse Drive, Waltham, Massachusetts 02451, United States.
  • Pontz T; Oncology Innovative Medicines Unit, AstraZeneca R&D , 35 Gatehouse Drive, Waltham, Massachusetts 02451, United States.
  • Ye Q; Oncology Innovative Medicines Unit, AstraZeneca R&D , 35 Gatehouse Drive, Waltham, Massachusetts 02451, United States.
  • Holdgate GA; Structure & Biophysics, Discovery Sciences, AstraZeneca R&D , Darwin Building, 310 Cambridge Science Park, Milton Road, Cambridge, CB4 0WG, U.K.
  • Snow L; Structure & Biophysics, Discovery Sciences, AstraZeneca R&D , Darwin Building, 310 Cambridge Science Park, Milton Road, Cambridge, CB4 0WG, U.K.
  • O'Connell N; Structure & Biophysics, Discovery Sciences, AstraZeneca R&D , 35 Gatehouse Drive, Waltham, Massachusetts 02451, United States.
  • Ferguson AD; Structure & Biophysics, Discovery Sciences, AstraZeneca R&D , 35 Gatehouse Drive, Waltham, Massachusetts 02451, United States.
ACS Med Chem Lett ; 7(3): 300-5, 2016 Mar 10.
Article in En | MEDLINE | ID: mdl-26985319

Full text: 1 Collection: 01-internacional Database: MEDLINE Language: En Journal: ACS Med Chem Lett Year: 2016 Document type: Article Affiliation country: United States Country of publication: United States

Full text: 1 Collection: 01-internacional Database: MEDLINE Language: En Journal: ACS Med Chem Lett Year: 2016 Document type: Article Affiliation country: United States Country of publication: United States