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Novel BQCA- and TBPB-Derived M1 Receptor Hybrid Ligands: Orthosteric Carbachol Differentially Regulates Partial Agonism.
Schramm, Simon; Agnetta, Luca; Bermudez, Marcel; Gerwe, Hubert; Irmen, Matthias; Holze, Janine; Littmann, Timo; Wolber, Gerhard; Tränkle, Christian; Decker, Michael.
Affiliation
  • Schramm S; Pharmazeutische und Medizinische Chemie, Institut für Pharmazie und Lebensmittelchemie, Julius-Maximilians-Universität Würzburg, Am Hubland, 97074, Würzburg, Germany.
  • Agnetta L; Pharmazeutische und Medizinische Chemie, Institut für Pharmazie und Lebensmittelchemie, Julius-Maximilians-Universität Würzburg, Am Hubland, 97074, Würzburg, Germany.
  • Bermudez M; Institute of Pharmacy, Freie Universität Berlin, Königin-Luise-Strasse 2+4, 14195, Berlin, Germany.
  • Gerwe H; Pharmazeutische und Medizinische Chemie, Institut für Pharmazie und Lebensmittelchemie, Julius-Maximilians-Universität Würzburg, Am Hubland, 97074, Würzburg, Germany.
  • Irmen M; Pharmacology and Toxicology, Institute of Pharmacy, University of Bonn, Gerhard-Domagk-Strasse 3, 53121, Bonn, Germany.
  • Holze J; Pharmacology and Toxicology, Institute of Pharmacy, University of Bonn, Gerhard-Domagk-Strasse 3, 53121, Bonn, Germany.
  • Littmann T; Institute of Pharmacy, University of Regensburg, 93053, Regensburg, Germany.
  • Wolber G; Institute of Pharmacy, Freie Universität Berlin, Königin-Luise-Strasse 2+4, 14195, Berlin, Germany.
  • Tränkle C; Pharmacology and Toxicology, Institute of Pharmacy, University of Bonn, Gerhard-Domagk-Strasse 3, 53121, Bonn, Germany.
  • Decker M; Pharmazeutische und Medizinische Chemie, Institut für Pharmazie und Lebensmittelchemie, Julius-Maximilians-Universität Würzburg, Am Hubland, 97074, Würzburg, Germany.
ChemMedChem ; 14(14): 1349-1358, 2019 07 17.
Article in En | MEDLINE | ID: mdl-31166078

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Piperidines / Quinolines / Benzimidazoles / Carbachol / Receptor, Muscarinic M1 Limits: Humans Language: En Journal: ChemMedChem Journal subject: FARMACOLOGIA / QUIMICA Year: 2019 Document type: Article Affiliation country: Germany Country of publication: Germany

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Piperidines / Quinolines / Benzimidazoles / Carbachol / Receptor, Muscarinic M1 Limits: Humans Language: En Journal: ChemMedChem Journal subject: FARMACOLOGIA / QUIMICA Year: 2019 Document type: Article Affiliation country: Germany Country of publication: Germany