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Mechanistic insights into the activation of ester prodrugs of 666-15.
Xie, Fuchun; Martín-Acosta, Pedro; Li, Bingbing X; Xiao, Xiangshu.
Affiliation
  • Xie F; Program in Chemical Biology, Department of Chemical Physiology and Biochemistry, 3181 SW Sam Jackson Park Road, Portland, OR 97239, United States.
  • Martín-Acosta P; Program in Chemical Biology, Department of Chemical Physiology and Biochemistry, 3181 SW Sam Jackson Park Road, Portland, OR 97239, United States.
  • Li BX; Program in Chemical Biology, Department of Chemical Physiology and Biochemistry, 3181 SW Sam Jackson Park Road, Portland, OR 97239, United States.
  • Xiao X; Program in Chemical Biology, Department of Chemical Physiology and Biochemistry, 3181 SW Sam Jackson Park Road, Portland, OR 97239, United States; Knight Cancer Institute, Oregon Health & Science University, 3181 SW Sam Jackson Park Road, Portland, OR 97239, United States. Electronic address: xi
Bioorg Med Chem Lett ; 30(19): 127455, 2020 10 01.
Article in En | MEDLINE | ID: mdl-32730943

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Prodrugs / Cyclic AMP Response Element-Binding Protein / Esters / Anilides / Naphthalenes Limits: Humans Language: En Journal: Bioorg Med Chem Lett Journal subject: BIOQUIMICA / QUIMICA Year: 2020 Document type: Article Affiliation country: United States Country of publication: United kingdom

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Prodrugs / Cyclic AMP Response Element-Binding Protein / Esters / Anilides / Naphthalenes Limits: Humans Language: En Journal: Bioorg Med Chem Lett Journal subject: BIOQUIMICA / QUIMICA Year: 2020 Document type: Article Affiliation country: United States Country of publication: United kingdom