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Picking the tyrosine-lock: chemical synthesis of the tyrosyl-DNA phosphodiesterase I inhibitor recifin A and analogues.
Smallwood, Taylor B; Krumpe, Lauren R H; Payne, Colton D; Klein, Victoria G; O'Keefe, Barry R; Clark, Richard J; Schroeder, Christina I; Rosengren, K Johan.
Affiliation
  • Smallwood TB; The University of Queensland, School of Biomedical Sciences Brisbane QLD 4072 Australia richard.clark@uq.edu.au j.rosengren@uq.edu.au.
  • Krumpe LRH; Molecular Targets Program, Centre for Cancer Research, National Cancer Institute, National Institute of Health Frederick MD 21702 USA.
  • Payne CD; The University of Queensland, School of Biomedical Sciences Brisbane QLD 4072 Australia richard.clark@uq.edu.au j.rosengren@uq.edu.au.
  • Klein VG; Chemical Biology Laboratory, Centre for Cancer Research, National Cancer Institute, National Institute of Health Frederick MD 21702 USA.
  • O'Keefe BR; Molecular Targets Program, Centre for Cancer Research, National Cancer Institute, National Institute of Health Frederick MD 21702 USA.
  • Clark RJ; Natural Products Branch, Centre for Cancer Research, National Cancer Institute, National Institute of Health Frederick MD 21702 USA.
  • Schroeder CI; The University of Queensland, School of Biomedical Sciences Brisbane QLD 4072 Australia richard.clark@uq.edu.au j.rosengren@uq.edu.au.
  • Rosengren KJ; Chemical Biology Laboratory, Centre for Cancer Research, National Cancer Institute, National Institute of Health Frederick MD 21702 USA.
Chem Sci ; 15(33): 13227-13233, 2024 Aug 22.
Article in En | MEDLINE | ID: mdl-39183914

Full text: 1 Collection: 01-internacional Database: MEDLINE Language: En Journal: Chem Sci Year: 2024 Document type: Article Country of publication: United kingdom

Full text: 1 Collection: 01-internacional Database: MEDLINE Language: En Journal: Chem Sci Year: 2024 Document type: Article Country of publication: United kingdom