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Phenyl Benzenesulfonylhydrazides Exhibit Selective Indoleamine 2,3-Dioxygenase Inhibition with Potent in Vivo Pharmacodynamic Activity and Antitumor Efficacy.
Lin, Shu-Yu; Yeh, Teng-Kuang; Kuo, Ching-Chuan; Song, Jen-Shin; Cheng, Ming-Fu; Liao, Fang-Yu; Chao, Min-Wu; Huang, Han-Li; Chen, Yi-Lin; Yang, Chun-Yu; Wu, Mine-Hsine; Hsieh, Chia-Ling; Hsiao, Wenchi; Peng, Yi-Hui; Wu, Jian-Sung; Lin, Li-Mei; Sun, Manwu; Chao, Yu-Sheng; Shih, Chuan; Wu, Su-Ying; Pan, Shiow-Lin; Hung, Ming-Shiu; Ueng, Shau-Hua.
Afiliación
  • Lin SY; Institute of Biotechnology and Pharmaceutical Research, National Health Research Institutes , Miaoli County 35053, Taiwan.
  • Yeh TK; Institute of Biotechnology and Pharmaceutical Research, National Health Research Institutes , Miaoli County 35053, Taiwan.
  • Kuo CC; Institute of Biotechnology and Pharmaceutical Research, National Health Research Institutes , Miaoli County 35053, Taiwan.
  • Song JS; Institute of Biotechnology and Pharmaceutical Research, National Health Research Institutes , Miaoli County 35053, Taiwan.
  • Cheng MF; Institute of Biotechnology and Pharmaceutical Research, National Health Research Institutes , Miaoli County 35053, Taiwan.
  • Liao FY; Institute of Biotechnology and Pharmaceutical Research, National Health Research Institutes , Miaoli County 35053, Taiwan.
  • Chao MW; The Ph.D. Program for Cancer Biology and Drug Discovery, College of Medical Science and Technology, Taipei Medical University , No. 250, Wu-Hsing Street, Taipei 11031, Taiwan.
  • Huang HL; The Ph.D. Program for Cancer Biology and Drug Discovery, College of Medical Science and Technology, Taipei Medical University , No. 250, Wu-Hsing Street, Taipei 11031, Taiwan.
  • Chen YL; The Ph.D. Program for Cancer Biology and Drug Discovery, College of Medical Science and Technology, Taipei Medical University , No. 250, Wu-Hsing Street, Taipei 11031, Taiwan.
  • Yang CY; Institute of Biotechnology and Pharmaceutical Research, National Health Research Institutes , Miaoli County 35053, Taiwan.
  • Wu MH; Institute of Biotechnology and Pharmaceutical Research, National Health Research Institutes , Miaoli County 35053, Taiwan.
  • Hsieh CL; Institute of Biotechnology and Pharmaceutical Research, National Health Research Institutes , Miaoli County 35053, Taiwan.
  • Hsiao W; Institute of Biotechnology and Pharmaceutical Research, National Health Research Institutes , Miaoli County 35053, Taiwan.
  • Peng YH; Institute of Biotechnology and Pharmaceutical Research, National Health Research Institutes , Miaoli County 35053, Taiwan.
  • Wu JS; Institute of Biotechnology and Pharmaceutical Research, National Health Research Institutes , Miaoli County 35053, Taiwan.
  • Lin LM; Institute of Biotechnology and Pharmaceutical Research, National Health Research Institutes , Miaoli County 35053, Taiwan.
  • Sun M; Institute of Biotechnology and Pharmaceutical Research, National Health Research Institutes , Miaoli County 35053, Taiwan.
  • Chao YS; Institute of Biotechnology and Pharmaceutical Research, National Health Research Institutes , Miaoli County 35053, Taiwan.
  • Shih C; Institute of Biotechnology and Pharmaceutical Research, National Health Research Institutes , Miaoli County 35053, Taiwan.
  • Wu SY; Institute of Biotechnology and Pharmaceutical Research, National Health Research Institutes , Miaoli County 35053, Taiwan.
  • Pan SL; The Ph.D. Program for Cancer Biology and Drug Discovery, College of Medical Science and Technology, Taipei Medical University , No. 250, Wu-Hsing Street, Taipei 11031, Taiwan.
  • Hung MS; Institute of Biotechnology and Pharmaceutical Research, National Health Research Institutes , Miaoli County 35053, Taiwan.
  • Ueng SH; Institute of Biotechnology and Pharmaceutical Research, National Health Research Institutes , Miaoli County 35053, Taiwan.
J Med Chem ; 59(1): 419-30, 2016 Jan 14.
Article en En | MEDLINE | ID: mdl-26653033

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Inhibidores Enzimáticos / Indolamina-Pirrol 2,3,-Dioxigenasa / Antineoplásicos Límite: Animals / Humans / Male Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2016 Tipo del documento: Article País de afiliación: Taiwán Pais de publicación: Estados Unidos

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Inhibidores Enzimáticos / Indolamina-Pirrol 2,3,-Dioxigenasa / Antineoplásicos Límite: Animals / Humans / Male Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2016 Tipo del documento: Article País de afiliación: Taiwán Pais de publicación: Estados Unidos