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Design, Synthesis and Biological Evaluation of Novel 1,2,5-Oxadiazol-3- Carboximidamide Derivatives as Indoleamine 2, 3-Dioxygenase 1 (IDO1) Inhibitors.
Xia, Zhifeng; Nan, Yanyang; Liu, Chang; Lin, Guangyu; Gu, Kedan; Chen, Cheng; Zhao, Weili; Ju, Dianwen; Dong, Xiaochun.
Afiliación
  • Xia Z; Department of Medicinal Chemistry, School of Pharmacy, Fudan University, Shanghai, 201203, China.
  • Nan Y; Department of Microbiological and Biochemical Pharmacy, School of Pharmacy, Fudan University, Shanghai, 201203, China.
  • Liu C; Department of Medicinal Chemistry, School of Pharmacy, Fudan University, Shanghai, 201203, China.
  • Lin G; Department of Medicinal Chemistry, School of Pharmacy, Fudan University, Shanghai, 201203, China.
  • Gu K; Department of Medicinal Chemistry, School of Pharmacy, Fudan University, Shanghai, 201203, China.
  • Chen C; Department of Medicinal Chemistry, School of Pharmacy, Fudan University, Shanghai, 201203, China.
  • Zhao W; Department of Medicinal Chemistry, School of Pharmacy, Fudan University, Shanghai, 201203, China.
  • Ju D; Department of Microbiological and Biochemical Pharmacy, School of Pharmacy, Fudan University, Shanghai, 201203, China.
  • Dong X; Department of Medicinal Chemistry, School of Pharmacy, Fudan University, Shanghai, 201203, China.
Anticancer Agents Med Chem ; 20(13): 1592-1603, 2020.
Article en En | MEDLINE | ID: mdl-32496990

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Oxadiazoles / Diseño de Fármacos / Carcinoma Pulmonar de Lewis / Inhibidores Enzimáticos / Indolamina-Pirrol 2,3,-Dioxigenasa / Antineoplásicos Límite: Animals / Humans Idioma: En Revista: Anticancer Agents Med Chem Asunto de la revista: ANTINEOPLASICOS / QUIMICA Año: 2020 Tipo del documento: Article País de afiliación: China

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Oxadiazoles / Diseño de Fármacos / Carcinoma Pulmonar de Lewis / Inhibidores Enzimáticos / Indolamina-Pirrol 2,3,-Dioxigenasa / Antineoplásicos Límite: Animals / Humans Idioma: En Revista: Anticancer Agents Med Chem Asunto de la revista: ANTINEOPLASICOS / QUIMICA Año: 2020 Tipo del documento: Article País de afiliación: China