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A site-moiety map and virtual screening approach for discovery of novel 5-LOX inhibitors.
Hsu, Kai-Cheng; HuangFu, Wei-Chun; Lin, Tony Eight; Chao, Min-Wu; Sung, Tzu-Ying; Chen, Yi-Ying; Pan, Shiow-Lin; Lee, Jih-Chin; Tzou, Shey-Cherng; Sun, Chung-Ming; Yang, Jinn-Moon.
Afiliación
  • Hsu KC; Graduate Institute of Cancer Biology and Drug Discovery, College of Medical Science and Technology, Taipei Medical University, Taipei, Taiwan.
  • HuangFu WC; Ph.D. Program for Cancer Molecular Biology and Drug Discovery, College of Medical Science and Technology, Taipei Medical University, Taipei, Taiwan.
  • Lin TE; Ph.D. Program in Biotechnology Research and Development, College of Pharmacy, Taipei Medical University, Taipei, Taiwan.
  • Chao MW; Biomedical Commercialization Center, Taipei Medical University, Taipei, Taiwan.
  • Sung TY; Graduate Institute of Cancer Biology and Drug Discovery, College of Medical Science and Technology, Taipei Medical University, Taipei, Taiwan.
  • Chen YY; Ph.D. Program for Cancer Molecular Biology and Drug Discovery, College of Medical Science and Technology, Taipei Medical University, Taipei, Taiwan.
  • Pan SL; Ph.D. Program in Biotechnology Research and Development, College of Pharmacy, Taipei Medical University, Taipei, Taiwan.
  • Lee JC; Graduate Institute of Cancer Biology and Drug Discovery, College of Medical Science and Technology, Taipei Medical University, Taipei, Taiwan.
  • Tzou SC; Ph.D. Program for Cancer Molecular Biology and Drug Discovery, College of Medical Science and Technology, Taipei Medical University, Taipei, Taiwan.
  • Sun CM; Graduate Institute of Cancer Biology and Drug Discovery, College of Medical Science and Technology, Taipei Medical University, Taipei, Taiwan.
  • Yang JM; Institute of Bioinformatics and Systems Biology, National Chiao Tung University, Hsinchu, Taiwan.
Sci Rep ; 10(1): 10510, 2020 06 29.
Article en En | MEDLINE | ID: mdl-32601404

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Inhibidores de la Lipooxigenasa / Descubrimiento de Drogas / Inflamación / Antiinflamatorios Tipo de estudio: Diagnostic_studies / Screening_studies Límite: Humans Idioma: En Revista: Sci Rep Año: 2020 Tipo del documento: Article País de afiliación: Taiwán Pais de publicación: Reino Unido

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Inhibidores de la Lipooxigenasa / Descubrimiento de Drogas / Inflamación / Antiinflamatorios Tipo de estudio: Diagnostic_studies / Screening_studies Límite: Humans Idioma: En Revista: Sci Rep Año: 2020 Tipo del documento: Article País de afiliación: Taiwán Pais de publicación: Reino Unido