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Covalent Inhibition of Wild-Type HIV-1 Reverse Transcriptase Using a Fluorosulfate Warhead.
Ippolito, Joseph A; Niu, Haichan; Bertoletti, Nicole; Carter, Zachary J; Jin, Shengyan; Spasov, Krasimir A; Cisneros, José A; Valhondo, Margarita; Cutrona, Kara J; Anderson, Karen S; Jorgensen, William L.
Afiliación
  • Ippolito JA; Department of Chemistry, Yale University, New Haven, Connecticut 06520-8107, United States.
  • Niu H; Department of Pharmacology, Yale University School of Medicine, New Haven, Connecticut 06520-8066, United States.
  • Bertoletti N; Department of Chemistry, Yale University, New Haven, Connecticut 06520-8107, United States.
  • Carter ZJ; Department of Pharmacology, Yale University School of Medicine, New Haven, Connecticut 06520-8066, United States.
  • Jin S; Department of Chemistry, Yale University, New Haven, Connecticut 06520-8107, United States.
  • Spasov KA; Department of Pharmacology, Yale University School of Medicine, New Haven, Connecticut 06520-8066, United States.
  • Cisneros JA; Department of Pharmacology, Yale University School of Medicine, New Haven, Connecticut 06520-8066, United States.
  • Valhondo M; Department of Chemistry, Yale University, New Haven, Connecticut 06520-8107, United States.
  • Cutrona KJ; Department of Chemistry, Yale University, New Haven, Connecticut 06520-8107, United States.
  • Anderson KS; Department of Chemistry, Yale University, New Haven, Connecticut 06520-8107, United States.
  • Jorgensen WL; Department of Pharmacology, Yale University School of Medicine, New Haven, Connecticut 06520-8066, United States.
ACS Med Chem Lett ; 12(2): 249-255, 2021 Feb 11.
Article en En | MEDLINE | ID: mdl-33603971

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Idioma: En Revista: ACS Med Chem Lett Año: 2021 Tipo del documento: Article País de afiliación: Estados Unidos Pais de publicación: Estados Unidos

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Idioma: En Revista: ACS Med Chem Lett Año: 2021 Tipo del documento: Article País de afiliación: Estados Unidos Pais de publicación: Estados Unidos