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Discovery, synthesis and exploration of N-benzylsulfonyl-2-phenylazepanes as inhibitors of Bim expression in a mouse embryonic fibroblast model.
Richards, Benjamin J; Glab, Jason A; Mbogo, George W; Dahanayake, Darani; Smith, Brian J; Puthalakath, Hamsa; Abbott, Belinda M.
Afiliación
  • Richards BJ; Department of Chemistry and Physics, La Trobe Institute for Molecular Science, La Trobe University, Melbourne, Victoria 3086, Australia.
  • Glab JA; Department of Biochemistry and Genetics, La Trobe Institute for Molecular Science, La Trobe University, Melbourne, Victoria 3086, Australia.
  • Mbogo GW; Department of Biochemistry and Genetics, La Trobe Institute for Molecular Science, La Trobe University, Melbourne, Victoria 3086, Australia.
  • Dahanayake D; Department of Chemistry and Physics, La Trobe Institute for Molecular Science, La Trobe University, Melbourne, Victoria 3086, Australia.
  • Smith BJ; Department of Chemistry and Physics, La Trobe Institute for Molecular Science, La Trobe University, Melbourne, Victoria 3086, Australia.
  • Puthalakath H; Department of Biochemistry and Genetics, La Trobe Institute for Molecular Science, La Trobe University, Melbourne, Victoria 3086, Australia.
  • Abbott BM; Department of Chemistry and Physics, La Trobe Institute for Molecular Science, La Trobe University, Melbourne, Victoria 3086, Australia. Electronic address: b.abbott@latrobe.edu.au.
Bioorg Chem ; 120: 105635, 2022 03.
Article en En | MEDLINE | ID: mdl-35124512

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Proteínas Proto-Oncogénicas / Insuficiencia Cardíaca Límite: Animals Idioma: En Revista: Bioorg Chem Año: 2022 Tipo del documento: Article País de afiliación: Australia Pais de publicación: Estados Unidos

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Proteínas Proto-Oncogénicas / Insuficiencia Cardíaca Límite: Animals Idioma: En Revista: Bioorg Chem Año: 2022 Tipo del documento: Article País de afiliación: Australia Pais de publicación: Estados Unidos