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A novel screening strategy to identify histone methyltransferase inhibitors reveals a crosstalk between DOT1L and CARM1.
Si, Yang; Bon, Corentin; Barbachowska, Magdalena; Cadet-Daniel, Veronique; Jallet, Corinne; Soresinetti, Laura; Boullé, Mikaël; Duchateau, Magalie; Matondo, Mariette; Agou, Fabrice; Halby, Ludovic; Arimondo, Paola B.
Afiliación
  • Si Y; Epigenetic Chemical Biology, Department of Structural Biology and Chemistry, Institut Pasteur, UMR3523 CNRS 75015 Paris France paola.arimondo@cnrs.fr.
  • Bon C; Epigenetic Chemical Biology, Department of Structural Biology and Chemistry, Institut Pasteur, UMR3523 CNRS 75015 Paris France paola.arimondo@cnrs.fr.
  • Barbachowska M; Ecole Doctorale MTCI, Université de Paris, Sorbonne Paris Cité Paris France.
  • Cadet-Daniel V; Epigenetic Chemical Biology, Department of Structural Biology and Chemistry, Institut Pasteur, UMR3523 CNRS 75015 Paris France paola.arimondo@cnrs.fr.
  • Jallet C; Ecole Doctorale MTCI, Université de Paris, Sorbonne Paris Cité Paris France.
  • Soresinetti L; Epigenetic Chemical Biology, Department of Structural Biology and Chemistry, Institut Pasteur, UMR3523 CNRS 75015 Paris France paola.arimondo@cnrs.fr.
  • Boullé M; Epigenetic Chemical Biology, Department of Structural Biology and Chemistry, Institut Pasteur, UMR3523 CNRS 75015 Paris France paola.arimondo@cnrs.fr.
  • Duchateau M; Epigenetic Chemical Biology, Department of Structural Biology and Chemistry, Institut Pasteur, UMR3523 CNRS 75015 Paris France paola.arimondo@cnrs.fr.
  • Matondo M; Chemogenomics and Biology Screening platform, Institut Pasteur 75015 Paris France.
  • Agou F; Proteomic Platform, Mass spectrometry for Biology, CNRS USR 2000, Institut Pasteur 75015 Paris France.
  • Halby L; Proteomic Platform, Mass spectrometry for Biology, CNRS USR 2000, Institut Pasteur 75015 Paris France.
  • Arimondo PB; Chemogenomics and Biology Screening platform, Institut Pasteur 75015 Paris France.
RSC Chem Biol ; 3(4): 456-467, 2022 Apr 06.
Article en En | MEDLINE | ID: mdl-35441144

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Tipo de estudio: Diagnostic_studies / Screening_studies Idioma: En Revista: RSC Chem Biol Año: 2022 Tipo del documento: Article

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Tipo de estudio: Diagnostic_studies / Screening_studies Idioma: En Revista: RSC Chem Biol Año: 2022 Tipo del documento: Article