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Evaluating the correlation of binding affinities between isothermal titration calorimetry and fragment molecular orbital method of estrogen receptor beta with diarylpropionitrile (DPN) or DPN derivatives.
Handa, Chiaki; Yamazaki, Yuki; Yonekubo, Shigeru; Furuya, Noritaka; Momose, Takaki; Ozawa, Tomonaga; Furuishi, Takayuki; Fukuzawa, Kaori; Yonemochi, Etsuo.
Afiliación
  • Handa C; Central Research Laboratory, Kissei Pharmaceutical Co., Ltd., 4365-1, Hotakakashiwabara, Azumino, Nagano 399-8304, Japan; School of Pharmacy and Pharmaceutical Sciences, Hoshi University, 2-4-41 Shinagawa, Tokyo 142-8501, Japan. Electronic address: chiaki_handa@pharm.kissei.co.jp.
  • Yamazaki Y; School of Pharmacy and Pharmaceutical Sciences, Hoshi University, 2-4-41 Shinagawa, Tokyo 142-8501, Japan.
  • Yonekubo S; Central Research Laboratory, Kissei Pharmaceutical Co., Ltd., 4365-1, Hotakakashiwabara, Azumino, Nagano 399-8304, Japan.
  • Furuya N; Central Research Laboratory, Kissei Pharmaceutical Co., Ltd., 4365-1, Hotakakashiwabara, Azumino, Nagano 399-8304, Japan.
  • Momose T; Central Research Laboratory, Kissei Pharmaceutical Co., Ltd., 4365-1, Hotakakashiwabara, Azumino, Nagano 399-8304, Japan.
  • Ozawa T; Central Research Laboratory, Kissei Pharmaceutical Co., Ltd., 4365-1, Hotakakashiwabara, Azumino, Nagano 399-8304, Japan.
  • Furuishi T; School of Pharmacy and Pharmaceutical Sciences, Hoshi University, 2-4-41 Shinagawa, Tokyo 142-8501, Japan.
  • Fukuzawa K; Graduate School of Pharmaceutical Sciences, Osaka University, 1-6 Yamadaoka, Suita, Osaka 565-0871, Japan.
  • Yonemochi E; School of Pharmacy and Pharmaceutical Sciences, Hoshi University, 2-4-41 Shinagawa, Tokyo 142-8501, Japan.
J Steroid Biochem Mol Biol ; 222: 106152, 2022 09.
Article en En | MEDLINE | ID: mdl-35810932

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Receptor alfa de Estrógeno / Receptor beta de Estrógeno Idioma: En Revista: J Steroid Biochem Mol Biol Asunto de la revista: BIOLOGIA MOLECULAR / BIOQUIMICA Año: 2022 Tipo del documento: Article Pais de publicación: Reino Unido

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Receptor alfa de Estrógeno / Receptor beta de Estrógeno Idioma: En Revista: J Steroid Biochem Mol Biol Asunto de la revista: BIOLOGIA MOLECULAR / BIOQUIMICA Año: 2022 Tipo del documento: Article Pais de publicación: Reino Unido