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Discovery of small molecule FLT3 inhibitors that are able to overcome drug-resistant mutations.
Zhang, Guo; Zhang, Wenqing; Shen, Chenjian; Nan, Jinshan; Chen, Ming; Lai, Shusheng; Zhong, Jiemin; Li, Bolin; Wang, Tianqi; Wang, Yifei; Yang, Shengyong; Li, Linli.
Afiliação
  • Zhang G; State Key Laboratory of Biotherapy and Cancer Center, West China Hospital, Sichuan University, Sichuan 610041, China.
  • Zhang W; Key Laboratory of Drug Targeting and Drug Delivery System of Ministry of Education, West China School of Pharmacy, Sichuan University, Sichuan 610041, China.
  • Shen C; State Key Laboratory of Biotherapy and Cancer Center, West China Hospital, Sichuan University, Sichuan 610041, China.
  • Nan J; State Key Laboratory of Biotherapy and Cancer Center, West China Hospital, Sichuan University, Sichuan 610041, China.
  • Chen M; Guangxi Wuzhou Pharmaceutical Co. Ltd, Wuzhou, Guangxi 543000, China.
  • Lai S; Guangxi Wuzhou Pharmaceutical Co. Ltd, Wuzhou, Guangxi 543000, China.
  • Zhong J; Guangxi Wuzhou Pharmaceutical Co. Ltd, Wuzhou, Guangxi 543000, China.
  • Li B; Guangxi Wuzhou Pharmaceutical Co. Ltd, Wuzhou, Guangxi 543000, China.
  • Wang T; State Key Laboratory of Biotherapy and Cancer Center, West China Hospital, Sichuan University, Sichuan 610041, China.
  • Wang Y; Key Laboratory of Drug Targeting and Drug Delivery System of Ministry of Education, West China School of Pharmacy, Sichuan University, Sichuan 610041, China.
  • Yang S; State Key Laboratory of Biotherapy and Cancer Center, West China Hospital, Sichuan University, Sichuan 610041, China.
  • Li L; Key Laboratory of Drug Targeting and Drug Delivery System of Ministry of Education, West China School of Pharmacy, Sichuan University, Sichuan 610041, China. Electronic address: lilinli@scu.edu.cn.
Bioorg Med Chem Lett ; 30(22): 127532, 2020 11 15.
Article em En | MEDLINE | ID: mdl-32891702

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Ureia / Resistencia a Medicamentos Antineoplásicos / Inibidores de Proteínas Quinases / Tirosina Quinase 3 Semelhante a fms / Bibliotecas de Moléculas Pequenas / Descoberta de Drogas Limite: Humans Idioma: En Revista: Bioorg Med Chem Lett Assunto da revista: BIOQUIMICA / QUIMICA Ano de publicação: 2020 Tipo de documento: Article País de afiliação: China País de publicação: Reino Unido

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Ureia / Resistencia a Medicamentos Antineoplásicos / Inibidores de Proteínas Quinases / Tirosina Quinase 3 Semelhante a fms / Bibliotecas de Moléculas Pequenas / Descoberta de Drogas Limite: Humans Idioma: En Revista: Bioorg Med Chem Lett Assunto da revista: BIOQUIMICA / QUIMICA Ano de publicação: 2020 Tipo de documento: Article País de afiliação: China País de publicação: Reino Unido