Folate receptor-mediated antitumor drugs / 药学学报
Acta Pharmaceutica Sinica
; (12): 109-114, 2009.
Article
em Zh
| WPRIM
| ID: wpr-232588
Biblioteca responsável:
WPRO
ABSTRACT
Folate receptor (FR) is over-expressed in a variety of human cancers and it is seldom expressed or found in normal tissues. Therefore, folate receptor-mediated antitumor drugs can be targeted specially to the FR-positive tumor cells. This strategy improves the selectivity of drugs which may destroy the normal tissues in traditional chemotherapeutics. This review provides the delivery mechanism of FR-mediated antitumor drugs and highlights the novel folate-drug conjugates and their activities.
Texto completo:
1
Base de dados:
WPRIM
Assunto principal:
Patologia
/
Farmacologia
/
Portadores de Fármacos
/
Proteínas de Transporte
/
Química
/
Sistemas de Liberação de Medicamentos
/
Receptores de Superfície Celular
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Linhagem Celular Tumoral
/
Receptores de Folato com Âncoras de GPI
/
Ácido Fólico
Limite:
Animals
/
Humans
Idioma:
Zh
Revista:
Acta Pharmaceutica Sinica
Ano de publicação:
2009
Tipo de documento:
Article